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4-(4-chlorophenyl)-N-[(2,4-dihydroxyphenyl)methyl]butanamide
N-cyclopropyl-3-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
N-(2,4-dimethoxyphenyl)-3-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}propanamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(4-chloro-1H-pyrazol-1-yl)propan-1-one
ethyl 1-[6-(1-benzothiophen-3-yl)-3-(4-formylpiperazine-1-carbonyl)pyridin-2-yl]piperidine-3-carboxylate
1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperidin-4-amine
methyl (2S)-1-({4-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)pyrrolidine-2-carboxylate
(3aR,5S,6S,7aS)-5,6-dihydroxy-N-(naphthalen-2-yl)-octahydro-1H-isoindole-2-carboxamide
[2-(1,3-benzothiazol-2-yl)ethyl](benzylsulfamoyl)amine
2-(5,7-dimethoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)benzonitrile
2-{4-[1-(pyridin-3-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxy}-1-(pyrrolidin-1-yl)ethan-1-one
(2R,3S,6R)-5-(2-cyclopropylpyrimidine-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{1-azabicyclo[2.2.2]octan-3-yl}-N-(pyridin-3-ylmethyl)-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
1-[(5-methylpyrazin-2-yl)methyl]-3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]urea
5-oxo-1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
(3R)-3-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[2-(1,3-thiazol-4-yl)ethyl]amine
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(oxane-2-carbonyl)piperidine-4-carboxylic acid
N-{2-[7-(naphthalen-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}pyridine-3-carboxamide
3-{2-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]ethyl}-1H-indole
1-[(2,6-difluorophenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
4-(4-fluorophenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-4-oxobutanamide
2-[4-(5-{[(3-fluorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]-N,N-dimethylacetamide
2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}acetamide
{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-benzamido-1-(furan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1S,5R)-3-[4-methyl-6-(methylamino)pyrimidin-2-yl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1-ethyl-1H-indazol-3-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-(2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-6-methyl-2,3-dihydropyridazin-3-one
3-[benzyl(1,3-thiazol-2-ylmethyl)amino]propane-1,2-diol
2-methyl-5-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrimidine
(1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)methanol
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)pyrrolidine-3-carboxylic acid
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(5-methyl-1H-pyrazol-1-yl)acetamide
2-(pyridin-2-ylsulfanyl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
1-[(2-fluorophenyl)methyl]-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
5-cyclopropyl-N-(2-methoxyethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-methyl-1H-pyrazole-4-carboxamide
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
5-(2,6-dimethoxypyrimidin-4-yl)quinoline
8-[6-(morpholin-4-yl)pyrimidin-4-yl]quinoline
3-(hydroxymethyl)-1-(2-phenoxybenzoyl)piperidin-3-ol
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidine-4-carboxamide
N,N-dimethyl-3-[2-({[(5-methylpyrazin-2-yl)methyl]carbamoyl}amino)phenyl]propanamide
3-hexyl-8-[2-(methylamino)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methyl-N-{[4-(piperidine-1-carbonyl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-[2-(methylsulfanyl)acetyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]acetamide