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3-cyclopropyl-6-(4-methoxy-3,5-dimethylphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-(2H-1,3-benzodioxol-5-yl)-N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}acetamide
1-methyl-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2,5-dimethyl-N-[3-(phenylsulfanyl)propyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
methyl 6-{[benzyl(methyl)amino]methyl}-3-(3-methylbenzamido)thieno[2,3-b]pyridine-2-carboxylate
2-ethyl-8-[6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-methyl-2-oxo-8-[3-(pyridin-4-yl)propanoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
2-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-4,5,6,7-tetrahydro-1,3-benzothiazole
3-(1-{[5-(3-hydroxypropanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperidin-4-yl)-1,3-oxazolidin-2-one
N,4-dimethyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-oxazole-5-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3-phenyl-1,2-oxazole-5-carboxamide
(4aS,8aR)-6-[2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)acetyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
3-(5-fluoro-2-methoxybenzoyl)-1-(1H-pyrazol-3-ylmethyl)piperidine
5-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)imidazolidine-2,4-dione
ethyl 2-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(thiophen-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-[(2,4-difluorophenyl)methyl]-3-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]urea
1-(oxane-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}quinoline-8-sulfonamide
2-amino-N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-methoxy-2-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1H-indole
3-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-phenyl-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
1-[(4aS,8aR)-6-acetyl-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
6-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-N-cyclopropyl-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-{[3-(2-methoxyethyl)-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[1-(thiophen-2-yl)ethyl]urea
5-[2-(ethylamino)ethyl]-1-[(1R)-1-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
2-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decane
1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
(1R,3S)-3-methoxy-3-methyl-7-[6-(trifluoromethyl)pyridin-2-yl]-7-azaspiro[3.5]nonan-1-ol
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(pyridin-2-yl)propan-1-one
4-methoxy-N-({1-[3-(methylsulfanyl)propanoyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
2-[methyl({4-[4-(4-methylphenoxy)piperidine-1-carbonyl]phenyl})amino]ethan-1-ol
1,5-dimethyl-4-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-(2-methylphenoxy)-1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidine-4-carboxylic acid
1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methoxypropan-1-one
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-N-ethyl-N-methylpyrimidin-4-amine
8-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(2-hydroxyethyl)amino)ethan-1-ol
2-hydroxy-4-[2-(phenylsulfanyl)ethoxy]-5-(pyrimidin-5-yl)benzoic acid
8-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-cycloheptyl-N-[1-(6-methoxynaphthalen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-9-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-[2-(3,5-dimethoxyphenyl)ethyl]-3-(1-methylpiperidin-4-yl)propanamide
(4aR,8aR)-2-(5-phenyl-1,2,4-oxadiazol-3-yl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol