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1-{2-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
4-{1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}benzoic acid
(3aS,6aS)-2-methyl-5-{[4-(trifluoromethyl)phenyl]carbamoyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{methyl[(3-methyl-1H-indol-2-yl)methyl]amino}-1-(3-methylpiperidin-1-yl)propan-1-one
2-[(3,4-difluorophenyl)methyl]-8-[1-(hydroxymethyl)cyclopropanecarbonyl]-2,8-diazaspiro[4.5]decan-3-one
1-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-({7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
2-[2-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)phenoxy]acetic acid
N-[3-(3-ethylphenoxy)propyl]-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-amine
3-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-4-methyl-1,2,5-oxadiazole
3-(1H-imidazol-1-yl)-1-[4-(4-methoxyphenoxy)piperidin-1-yl]butan-1-one
2-methoxy-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyridine
2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
2-(2-methoxyethyl)-8-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(2E)-2-methylbut-2-en-1-yl]amine
4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-(2-methylphenyl)piperazin-2-one
N-(1-benzylpyrrolidin-3-yl)-3-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)propanamide
(2S,4R)-1-(oxan-4-yl)-N-(propan-2-yl)-4-[2-(pyridin-4-yl)acetamido]pyrrolidine-2-carboxamide
(4aR,8aS)-1-(pyridin-3-ylmethyl)-6-[2-(3,4,5-trimethoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-2-one
2-phenyl-1-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]ethan-1-one
(2S,4R)-1-[(3-hydroxy-4-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{[(3S,4S)-3-hydroxy-1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl]methyl}-2-methoxyacetamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl})amine
(3aR,6aR)-2-(cyclobutylmethyl)-5-(4-fluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3,5-dichloropyridin-4-yl)methyl]-4-(oxan-4-yl)piperazine
9-[(2S,3R)-2-amino-3-hydroxybutanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-propyl-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)thiophene-3-carboxamide
4-(5-methyl-1,2,4-oxadiazol-3-yl)-1-{[2-(methylsulfanyl)phenyl]methyl}piperidine
(2S,4S,5R)-4-{[2-(dimethylamino)ethyl]carbamoyl}-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
8-(1H-imidazol-2-ylmethyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
4-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
4-[(3,5-dichloropyridin-4-yl)methyl]-2-ethyl-1-(propan-2-yl)piperazine
3-ethyl-8-[(1-methyl-1H-indol-6-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[2-(4-{[2-(cyclopentyloxy)phenyl]methyl}morpholin-2-yl)ethyl]dimethylamine
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(propylsulfanyl)acetamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetamide
1-(4-{1-[2-(2-hydroxyethoxy)ethyl]-4-phenyl-1H-imidazol-5-yl}thiophen-2-yl)ethan-1-one
methyl (2S,4S)-1-[(3,4-difluorophenyl)methyl]-4-(furan-2-amido)pyrrolidine-2-carboxylate
2-{4-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-2-oxopiperazin-1-yl}benzonitrile
2-{4-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidine-1-carbonyl]phenoxy}acetamide
N-[4-(methylsulfanyl)phenyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-(4-{4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]butanoyl}morpholin-3-yl)acetic acid
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(furan-2-yl)ethane-1,2-dione
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[2-(5-methylthiophen-2-yl)ethyl]propanamide
1-(4-cyclohexylphenyl)-3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
3-[(3S,4R)-4-(morpholin-4-yl)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
(3S,9aR)-2,3-dimethyl-8-[(4-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione