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N-{[(2S,4S)-1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-fluoropyrrolidin-2-yl]methyl}cyclopropanecarboxamide
2-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(1H-1,2,4-triazol-3-yl)-N-[(3,4,5-trimethoxyphenyl)methyl]benzamide
2-[methyl(1-methylpiperidin-4-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
(2S,4R)-4-amino-1-[(6-ethoxypyridin-3-yl)methyl]-N-methylpyrrolidine-2-carboxamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)oxane-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
1-(7-methoxy-4-methylquinazolin-2-yl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]piperidine-4-carboxamide
5-(1H-indol-3-ylmethyl)-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(2-ethylbutyl)-8-[2-(ethylsulfanyl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{1-benzyl-4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(1S,3R)-3-amino-N-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)cyclopentane-1-carboxamide
5-({8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1-ethyl-1H-1,2,4-triazole
(1R,2s,3S,6R,7r,8S)-N-(pyridin-2-ylmethyl)-11,12-dioxatetracyclo[6.2.1.13,6.02,7]dodecane-2-carboxamide
1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(3R,4R)-1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-3,4-dimethylpyrrolidin-3-ol
3,5-dimethyl-6-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
5-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
(4aS,7aR)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]phenyl}formamido)-N-methylacetamide
1-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)-3-{2-oxo-2-[2-(pyridin-3-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
3-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}-N-[3-(hydroxymethyl)phenyl]benzamide
2-amino-4-(3-hydroxy-4-methoxyphenyl)-5-methyl-6-phenylpyridine-3-carbonitrile
5-(3-methyl-3-phenylpiperidine-1-carbonyl)-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
1-(2-amino-6-methylpyrimidin-4-yl)-4-(1H-1,3-benzodiazol-1-yl)piperidine-4-carboxylic acid
N-[2-(3-methoxyphenoxy)ethyl]-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-({5-[(5-chlorothiophen-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
3-[2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)acetamido]-N-(1,3-thiazol-2-yl)propanamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylpent-4-enamide
N-[(5-methoxy-1H-indol-2-yl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
7-[2-(5-chloro-6-methyl-1-benzofuran-3-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]-5-(morpholine-4-sulfonyl)benzoic acid
(1H-imidazol-2-ylmethyl)(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-{[1-(3-chloro-2-methylphenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1H-1,2,3,4-tetrazole
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
7-[(4-fluorophenyl)methyl]-2-(3-methyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(4aR,8aS)-1-{[4-(furan-2-yl)phenyl]methyl}-decahydro-1,6-naphthyridin-6-yl]ethan-1-one
3-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridin-2-amine
methyl[(1-methyl-1H-imidazol-5-yl)methyl]{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methyl-2-phenylpropanamide
3-[4-(dimethylamino)phenyl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]propanamide
N-{[7-(2,4-dimethylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-2-one
4-methyl-5-{3-[(E)-2-phenylethenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-thiazole
4-[(1R)-1-(4-fluorophenyl)ethyl]-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-(hydroxymethyl)pyridin-2-yl]phenol
3-{4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazin-1-yl}benzoic acid
N,2,6-trimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidine-4-carboxamide