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3,5-dimethyl-N-(3-methyl-1-{7-propyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)benzamide
N-[2-(2-chlorophenyl)ethyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
N-(2-{7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
N-benzyl-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4,4,4-trifluorobutan-1-one
N-cyclopropyl-4-{[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}benzamide
4-(8-methyl-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}quinolin-2-yl)piperazin-2-one
1-(2-methoxy-4-methylbenzoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
2-(2-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-amine
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-5-(methoxymethyl)furan-2-carboxamide
{[3-(2-ethylmorpholine-4-carbonyl)-1,2-oxazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
2-methyl-5-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
2-{4-chloro-2-[(1S,5S)-3,6-diazabicyclo[3.2.2]nonan-3-ylmethyl]phenoxy}acetic acid
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]morpholine-4-sulfonamide
(3S,4S)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(3-methoxyphenyl)piperidin-3-ol
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-(1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl)propanamide
4-cyclobutanecarbonyl-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(5-{1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
4-[({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]benzonitrile
5-(2,3-dimethoxyphenyl)-1H-indazol-3-amine
N,2,5-trimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1,3-thiazole-4-carboxamide
1-(2-methoxyethyl)-3-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-1-(pyridin-4-ylmethyl)urea
5-chloro-7-methoxy-N-[2-(pyrrolidin-1-yl)ethyl]-1-benzofuran-2-carboxamide
N-ethyl-N-(pyridin-4-ylmethyl)-1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-amine
5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-(2-phenylethyl)piperidin-3-ol
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1,2-oxazolidin-2-yl)propanamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-{2-[3-(dimethylamino)propyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-5,6-dimethylpyridine-3-carbonitrile
3-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-chloropyridine
N-methyl-N-(propan-2-yl)-2-(1,3-thiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-[(2,6-dimethoxyphenyl)methyl]-3H,4H-pyrido[2,3-d]pyrimidin-4-one
3-(3-hydroxy-1,2-oxazol-5-yl)-1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}propan-1-one
8-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-5-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}pyrimidin-2-amine
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyridine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methanol
N-(2-hydroxyethyl)-3-(3-methoxyphenyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-4-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
methyl (2S,4R)-4-(2-phenylbenzamido)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}pent-4-en-1-one
2-(3,4-dimethylphenyl)-1-[(3R,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-1-yl]ethan-1-one
N-methyl-5-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}furan-2-carboxamide
3-{2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
N-[2-(dimethylamino)-2-methylpropyl]-3-{[(4-fluorophenyl)methyl]sulfanyl}propanamide
2-{3-methyl-4-[(4-phenyl-1,4-diazepan-1-yl)methyl]-1H-pyrazol-1-yl}ethan-1-ol
N-(2-hydroxyethyl)-1-[1-(2-methylquinolin-4-yl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-6-[(3,5-dichloropyridin-4-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide