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(3R,4R)-3-cyclopropyl-1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-4-methylpyrrolidin-3-ol
5-{[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]methyl}-3-phenyl-1,2,4-oxadiazole
2-methyl-6-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]phenol
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(isoquinolin-5-ylmethyl)methylamine
N-ethyl-3,5,7-trimethyl-N-(oxan-2-ylmethyl)-1H-indole-2-carboxamide
(4-{[({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)(methyl)amino]methyl}oxan-4-yl)methanol
methyl 5-[2-methyl-2-(thiophen-2-ylformamido)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]propan-1-one
1-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
5-methanesulfonyl-4-(piperidin-3-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidin-2-amine
1-[(3-chloro-4-methoxyphenyl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
2-[4-(3-cyanopyrazin-2-yl)piperazin-1-yl]-N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
4-benzyl-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-2-one
(1R,3S)-3-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]cyclopentan-1-amine
2-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)quinoline
4-(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)-6-methylpyrimidin-2-amine
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[4-(1H-pyrazol-1-yl)phenyl]methyl})amine
3,3-dimethyl-1-[(3S,4R)-1-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]urea
2-[4-(3,4-dichlorophenyl)piperazin-1-yl]-N-methylpyridine-4-carboxamide
2-(5-acetylthiophen-3-yl)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
2-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
(1S,2R)-2-{[(2-fluoro-4-methoxyphenyl)methyl](methyl)amino}cyclohexan-1-ol
(4S)-3-{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
1-(5-chloro-2-methylphenyl)-4-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
4-(2-methoxynaphthalen-1-yl)-1-(oxolan-3-yl)-1H-1,2,3-triazole
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(morpholin-4-yl)ethane-1,2-dione
4-(4-fluorophenyl)-4-hydroxy-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
3-{2-[4-(3-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-4-[(3-fluorophenyl)methyl]piperazin-2-one
4-(cyclopropylmethyl)-1-[2-(2-methylphenyl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-methyl-3-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
1-[4-(benzyloxy)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-(1-ethyl-5-oxopyrrolidin-3-yl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}benzamide
N-[(1R,2R)-1-[(6-cyclopropylpyrimidin-4-yl)amino]-2,3-dihydro-1H-inden-2-yl]acetamide
2-(1,3-thiazol-2-ylmethyl)-9-oxa-2-azaspiro[5.5]undecane
2-(1H-pyrazol-1-yl)-1-[(1s,5s)-7,10-dimethyl-3,7,10-triazatricyclo[3.3.3.01,5]undecan-3-yl]butan-1-one
6-(cyclobutylamino)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
methyl 7-oxo-3-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetyl]-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-cyclopropyl-3-{5-[2-(3,4-dimethylphenoxy)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
2-(2,2-dimethyloxan-4-yl)-1-[2-(3-methoxyphenyl)ethyl]-1H-imidazole
2-({4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
2-methyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-phenylpiperazine-1-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)acetamide
3-{[2-(ethoxymethyl)pyrrolidin-1-yl]sulfonyl}-N,N-diethylbenzamide
2-(3-methoxyphenyl)-1-[(4-methoxypiperidin-1-yl)sulfonyl]piperidine
3-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-6-methoxy-1,4-dihydroquinolin-4-one
2-[2-(4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazol-1-yl)ethyl]pyridine
5-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-N-ethylpyrimidin-2-amine