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N-{[3-methyl-7-(3-methylbenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}methanesulfonamide
1-(diphenylmethyl)-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-{1-cyclohexyl-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}benzamide
N-(1-benzylpiperidin-4-yl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(2-methoxyethyl)-1-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-fluoro-5-sulfamoyl-N-[1-(thiophen-3-yl)propan-2-yl]benzamide
[(2S,6S)-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(1S,5R)-3-(6-fluoro-4-hydroxyquinoline-3-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-ethyl-3-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]benzamide
2-{2-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]ethoxy}ethan-1-ol
{4-[3-(1H-pyrazol-1-yl)benzoyl]morpholin-2-yl}methanamine
N-[(2R,3R)-1'-(2,3-dimethylbenzoyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-methylpyridin-2-amine
3-(2-{[4-(1,5-dimethyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)pyridine
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-4-phenyl-9-(4-propylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecane
1-(4-fluorophenyl)-4-[2-(pyrrolidin-3-yl)benzoyl]piperazine
1-[2-({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-4-ol
N-[(1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methyl]acetamide
(1,4-dioxan-2-ylmethyl)({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})methylamine
2-[(4aR,7aS)-6,6-dioxo-4-{2-[(propan-2-yl)carbamoyl]ethyl}-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
5-{[3-(3-ethylphenoxy)azetidin-1-yl]methyl}-2-methoxybenzoic acid
(3S,4R)-1-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
methyl 4-[6-amino-5-cyano-4-(3-hydroxy-4-methoxyphenyl)pyridin-2-yl]-5-methylfuran-2-carboxylate
N-cyclopropyl-2-(piperidin-1-yl)-N-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}acetamide
(2E)-1-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(pyridin-4-yl)prop-2-en-1-one
4,4,4-trifluoro-1-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}butan-1-one
3-(4-phenyl-1H-imidazol-5-yl)phenol
[(3R,4R)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
ethyl 4-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-(2-methoxyphenyl)-4-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)piperazine
4-(4-methanesulfonylphenyl)-2-methoxypyridine-3-carbonitrile
5-[1-(5-acetylthiophene-3-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
(1S,5R)-3-benzyl-6-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(4-{[4-(6-chloropyridazin-3-yl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
3-(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
2-methyl-6-(1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)pyrimidin-4-ol
3-[4-(5-benzyl-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1-methyl-1,4-dihydroquinolin-4-one
6-[(4-methoxy-2,5-dimethylphenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-methoxy-6-(prop-2-en-1-yl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]phenol
3-(3-fluorophenyl)-6-(furan-2-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
[3-({1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(3-methanesulfonamido-4-methoxyphenyl)urea
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
2-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidine-1-carbonyl]benzonitrile
6-tert-butyl-1-methyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-(2-fluoro-3-methoxyphenyl)pyridin-2-amine