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2-ethyl-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-[(2-methoxyphenyl)methyl]-6-methyl-1,4-dihydropyridin-4-one
1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-phenylazepane
1-phenyl-3-(propan-2-yl)-4-[2-(propan-2-yl)-1,3-oxazol-4-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(4-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}phenyl)methanol
2-(2,3-dimethoxyphenyl)-1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazole
9-(6-methylpyrimidin-4-yl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(furan-2-yl)ethyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-ethyl-1-(2-methoxy-5-sulfamoylbenzoyl)piperidine-3-carboxylic acid
2-acetyl-8-[2-(2,3-dimethylphenoxy)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(4-fluorophenoxymethyl)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
5-{7-methylpyrazolo[1,5-a]pyrimidin-6-yl}-3-(2-phenylethyl)-1H-1,2,4-triazole
3-(cyclohex-1-en-1-yl)-5-(cyclopropylsulfamoyl)benzoic acid
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamide
5-[(5-chloro-2,3-dimethoxyphenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{5-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]thiophen-2-yl}ethan-1-one
3-{2-[7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-6-methoxy-2,3-dihydro-1H-indol-2-one
4-(furan-3-carbonyl)-N-(2-methoxypyridin-3-yl)-1,4-diazepane-1-carboxamide
3-hydroxy-3-{[(1H-indol-2-ylmethyl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amine
9-(4-methylpyrimidine-5-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
4-methoxy-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
3-cyclopropyl-4-[(2,4-dichlorophenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(ethanesulfonyl)-2-(3-phenylpropyl)morpholine
2-amino-4-cyclopropyl-6-(3-fluoro-4-methoxyphenyl)pyridine-3-carbonitrile
2-ethyl-8-[2-hydroxy-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}({[4-(trifluoromethyl)phenyl]methyl})amine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-[2-(cyclohexylsulfanyl)ethyl]-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
N-[(5-methylfuran-2-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-(6-hydroxy-4-{[(1-methyl-1H-pyrazol-4-yl)carbamoyl]methyl}-1,4-diazepan-1-yl)propanoic acid
3-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-(2-methoxyethyl)-1-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(2,5-dimethoxyphenyl)pyridine-4-carbonitrile
N-({7-[(2E)-3-(2,4-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)ethane-1-sulfonamide
1,3-dimethyl-N-[2-(1-methylpiperidin-2-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
methyl 1-[(3R,5S)-5-(4-phenylpiperazine-1-carbonyl)-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-(2-{7-[(3-phenoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(1,3-oxazol-5-yl)benzamide
N-methyl-1-[3-(1H-pyrazol-1-yl)propyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
N-{1-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-2-methoxyacetamide
8-(2H-1,3-benzodioxol-5-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
3-methyl-1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)butan-1-one
(5S,9aS,9bS)-5-(furan-2-yl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-({4-[(3-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-4-ol
3-ethoxy-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-4-(prop-2-en-1-yloxy)benzamide
1-(4-{4-[({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)amino]piperidin-1-yl}benzoyl)piperidin-3-ol