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5-(4-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
methyl (2S,4R)-4-(4-fluorobenzamido)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxylate
8-[(3-chloro-4-fluorophenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{3-[(4-fluorophenyl)formamido]propanoyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
1-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)-2-(1H-indol-1-yl)ethan-1-one
6-methyl-5-{5-[2-(1H-1,2,4-triazol-3-yl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
N-(1-benzylpiperidin-4-yl)-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
N-methyl-5-[1-(2-methyl-1,8-naphthyridine-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
methyl (1R,5S,6R)-6-({4-[2-(1H-pyrrol-1-yl)ethyl]piperazin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane-3-carboxylate
N-ethyl-5-({2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)pyrimidin-2-amine
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
5-[(2-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
(2S,4R)-4-amino-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-N-methylpyrrolidine-2-carboxamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)propanamide
1-methyl-4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}piperazine
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
2,5-dimethyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrazolo[1,5-a]pyrimidin-7-amine
(2R)-1-({3-methoxy-4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-2-methylpiperazine
5-[(furan-2-ylmethyl)amino]-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(4-cyclopentylpyrimidin-2-yl)-1-oxa-7-azaspiro[3.5]nonane
(4aS,7aR)-1-(6-methylpyridine-2-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4S,4aS,8aS)-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-decahydroquinolin-4-ol
N-[3-(dimethylamino)propyl]-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
N-benzyl-5-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}pyrimidin-2-amine
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]benzamide
2-(1-cyclopentyl-4-{[5-(hydroxymethyl)furan-2-yl]methyl}piperazin-2-yl)ethan-1-ol
N-(2-methoxyethyl)-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-methyl-1-benzofuran-5-carboxamide
3-[(3S,4R)-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-1-(2-methylpropyl)piperidin-3-yl]-1-[4-(4-fluorophenyl)piperazin-1-yl]propan-1-one
N-[(3-chlorophenyl)methyl]-3-{1-[2-(furan-2-yl)-2-oxoacetyl]piperidin-4-yl}propanamide
4-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]oxy}-3-chloro-N-(2-methoxyethyl)benzamide
2-amino-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
3-{2-[(benzylsulfamoyl)amino]phenyl}-N,N-dimethylpropanamide
2,6-dimethyl-N-[(4-phenylmorpholin-2-yl)methyl]quinoline-4-carboxamide
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-(1-methoxybutan-2-yl)benzamide
[(2-butyl-1H-imidazol-4-yl)methyl](propyl)(pyridin-3-ylmethyl)amine
2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-N-(thiophen-3-ylmethyl)pyridin-2-amine
1-(2-methoxyethyl)-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}pyrrolidine-3-carboxamide
3-methyl-6-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}pyridazine
1-(furan-2-yl)-2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]ethane-1,2-dione
1-(3,3-diphenylpiperidin-1-yl)-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-[2-(1H-1,3-benzodiazol-2-yl)acetamido]-N-methyl-N-phenylbenzamide
3-{1-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
methyl 3-[(1-cycloheptylpiperidin-3-yl)carbamoyl]benzoate
N-[1-(1-acetylpiperidin-4-yl)-1H-pyrazol-5-yl]-4-phenylbutanamide
1-{3-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2-oxoazepan-3-yl)-3-(pyridin-4-yl)propanamide