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1-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
(3R,5S)-5-(3-fluorophenoxymethyl)-N-(2-methylpropyl)piperidine-3-carboxamide
2-[3-({[2-(azepan-1-yl)ethyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[2-(4-methoxyphenyl)ethyl]piperidine-4-carboxamide
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1H-pyrazole-4-carboxamide
1-cyclopropanecarbonyl-4-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}piperidine
4-benzyl-3-ethyl-1-hexanoyl-1,4-diazepan-5-one
1-benzyl-6-[(4-hydroxy-3-methoxyphenyl)methyl]-3-(2-methoxyphenyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-({8-[(4-ethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)oxolane-2-carboxamide
1-[2-(4-cyclopentylpiperazin-1-yl)ethyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3,4-dimethyl-N-[1-(pyridin-3-yl)pentyl]-5-sulfamoylbenzamide
3-benzyl-4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperazin-2-one
N-{[7-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
4-(9-methoxy-7-oxo-3-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl)piperazin-2-one
1-methyl-3-(propan-2-yl)-8-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({3-[4-methoxy-4-(prop-2-en-1-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
2-[5-(2-chlorophenyl)-1,2-oxazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2,7,8-trimethyl-4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}quinoline
N-(2-methoxyethyl)-1-{1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carboxamide
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(4-methoxybenzoyl)piperazine
3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-one
6-methyl-4-[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
7-(5-chloro-2-methoxyphenyl)-9-methoxy-4-(quinolin-8-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(1-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}pyrrolidin-2-yl)thiophene-2-carboxamide
4-(2,3-dimethyl-1H-indole-7-carbonyl)-1λ6-thiomorpholine-1,1-dione
1-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-4-[(2-methylphenyl)sulfanyl]piperidine
3-(2H-1,3-benzodioxol-5-yl)-5-[(2E)-3-phenylprop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-fluoro-N-(2-oxoazepan-3-yl)-5-sulfamoylbenzamide
3-ethyl-5-hydroxy-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]adamantane-1-carboxamide
N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-2-(1,2-oxazolidin-2-yl)pyridine
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(2-methoxyethyl)propanamide
1-[(2S,3R)-2-amino-3-hydroxybutanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-({1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)piperazin-2-one
4'-{[4-(propan-2-yl)phenyl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl 4-[5-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
(3E)-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pent-3-en-1-one
4-[1-(3-methoxypropanoyl)piperidin-3-yl]benzoic acid
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methoxyphenoxy)piperidine
2-{6,8-dioxo-2,7-diazaspiro[4.4]nonan-2-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(1R,5R)-6-(1H-imidazol-2-ylmethyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-2-carboxamide
1-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
(2R,3R)-1'-(3-methylbut-2-en-1-yl)-3-(thiomorpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(4-fluorophenyl)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}propanamide
(4-benzyl-1-methylpiperidin-4-yl)methanol
N-[1-(1-{[(pyrazin-2-yl)carbamoyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-8-{[3-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione