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N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidin-4-amine
2-methyl-6-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-[(diethylamino)methyl]-5-ethylfuran-2-carboxamide
3-(4-chlorophenyl)-5-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
N-[(3R,4S)-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
2-(2-methoxyethyl)-9-(4-methoxypyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-5-[4-(thian-4-yl)piperazine-1-carbonyl]pyrimidine
[(3-{[1-(3-chlorobenzoyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(pyrazin-2-ylmethyl)amine
3-[2-({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)ethyl]-1,3-oxazolidin-2-one
8-fluoro-N-[3-(2-methoxyphenyl)propyl]quinoline-2-carboxamide
1-[2-(4-fluorophenyl)morpholin-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-[4-(methylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-methyl-4-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]benzene-1-sulfonamide
5-(1-benzofuran-2-yl)-3-[4-(thiomorpholin-4-yl)piperidin-1-yl]-1,2,4-triazine
2-(dimethylamino)-7-(1-ethyl-3-methylpiperidine-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{4-[(5-cyano-1-methyl-1H-pyrrol-3-yl)methyl]piperazin-1-yl}-N-ethylacetamide
(1S,5R)-6-(ethanesulfonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
ethyl 4-[1-(2-methoxyethyl)-2,4-dioxo-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]piperidine-1-carboxylate
methyl 3-(2-methoxybenzamido)-5-{[2-(4-methoxyphenyl)acetamido]methyl}benzoate
1-ethyl-4-{[methyl({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
4-[(3-ethyl-1H-pyrazol-5-yl)methyl]-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{1-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
methyl (2S)-2-phenyl-2-{[2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazolin-4-yl]formamido}acetate
1-[2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-2-yl)ethyl]pyrrolidin-2-one
2-{4-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-5,6-dimethylthieno[2,3-d]pyrimidin-2-yl}ethan-1-amine
2-(5-ethoxyfuran-2-carbonyl)-8-methyl-2,8-diazaspiro[4.5]decane
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-cyclohexyl-1H-1,2,3-triazole-4-carboxamide
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-5-({pyrazolo[1,5-a]pyrimidin-2-ylformamido}methyl)benzoate
2-{1-benzyl-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
1-(1-benzofuran-5-ylmethyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepane
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-4-sulfamoylbutanamide
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-7-oxo-3-(thiophene-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl 4-[(2-{[(1,3-benzothiazol-2-ylmethyl)(methyl)amino]methyl}quinazolin-4-yl)amino]butanoate
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]but-3-en-1-one
[(5-fluoro-1H-indol-2-yl)methyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{2-[4-(1,2,5-thiadiazole-3-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-3-(1-methyl-1H-imidazol-2-yl)piperidine
4-acetamido-N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
4-{1-[(3R,5S)-5-(pyrrolidine-1-carbonyl)piperidine-3-carbonyl]piperidin-4-yl}pyrimidine
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2,5-dimethyl-3-(4-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
1-(2-chloro-3-methoxyphenyl)-3-[(3-propyl-1,2-oxazol-5-yl)methyl]urea
2-fluoro-6-{4-[1-(piperidin-1-yl)ethyl]phenyl}benzamide
N-[(4-methoxyphenyl)methyl]-N,4,6-trimethylpyrimidin-2-amine
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-(3-methyl-1H-1,2,4-triazol-5-yl)-1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
1-(1,4-dithiepan-6-yl)-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-({[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
N-[(3S)-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide