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N-(3,5-dimethoxyphenyl)-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine-1-carboxamide
1-{4-[3-(thiomorpholin-4-ylmethyl)phenoxy]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
2-({[2-(azepan-1-yl)ethyl](propan-2-yl)amino}methyl)pyridine-3-carboxylic acid
1-(1-methylpiperidin-4-yl)-4-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidine
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[(4-methoxyphenyl)methyl]piperidin-4-amine
(2S,4S)-4-(benzylamino)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
N-[(3S,4R)-4-(propan-2-yl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)pyrrolidin-3-yl]methanesulfonamide
N-[(3R)-piperidin-3-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
(3S,4R)-4-(4-fluorophenyl)-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidine-3-carboxylic acid
4-(1H-1,2,3,4-tetrazol-5-yloxy)-N-(thiophen-3-ylmethyl)aniline
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
1-{3-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]propyl}pyrrolidin-2-one
3-(3-fluoro-4-phenylbenzoyl)-1-(oxan-4-yl)piperidine
5-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-(2-methylpropyl)-1H-imidazole
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-(4-fluorophenyl)urea
(1S,4S)-5-(2,2-diphenylacetyl)-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
2-{4-[(4-acetyl-1,4-diazepan-1-yl)methyl]phenyl}-6-butyl-3,4-dihydropyrimidin-4-one
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)amine
3-(2-oxo-2-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}ethyl)-3,4-dihydroquinazolin-4-one
2-methyl-N-[(5-methylpyrazin-2-yl)methyl]-3-[(pyridin-2-ylmethyl)amino]benzamide
6-chloro-2-{1-[5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazin-3-yl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
4-(2-methoxyphenyl)-2-methyl-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperazine
2-oxo-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1-oxaspiro[4.4]nonane-4-carboxamide
1-ethyl-4-[2-(4-methylpiperidine-1-carbonyl)-2,3-dihydro-1H-inden-2-yl]piperazine
4-phenyl-1-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}azepane
1-[3-(3-methoxyphenoxy)azetidin-1-yl]-4-(morpholin-4-yl)pentan-1-one
(2E)-1-{4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
5-(4-methoxyphenyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)furan-2-carboxamide
methyl 2-{2-[1-cyclohexyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamido}acetate
[(1-cyclopentylpiperidin-4-yl)methyl][(5-methylfuran-2-yl)methyl](pyridin-3-ylmethyl)amine
(4aR,7aS)-1-ethyl-4-{2-[methyl(1-methylpiperidin-4-yl)amino]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}pyridine
1-(4-{[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-2-yl)ethan-1-one
methyl 3-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}benzoate
1-methyl-9-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]propanamide
(1R,5R)-N,N-dimethyl-6-(3-phenoxypropanoyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-(hydroxymethyl)-2-methyl-4-({methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amino}methyl)pyridin-3-ol
N-(4-{1-[1-(pyrazin-2-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
methyl 3-[(2,5-difluorophenyl)methyl]-9-[(4-fluorophenyl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{[1-ethyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
(1-methyl-1H-imidazol-2-yl)(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)methanol
N-{[2-(diethylamino)pyridin-3-yl]methyl}pyridine-3-carboxamide
(3S,4R)-1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
N3-benzyl-1-cyclopropyl-N5-[(3-fluorophenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-(3-chloro-1,2-oxazol-5-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
N-{1-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
4-(1-benzylpiperidin-4-yl)-1,4-oxazepan-6-ol
2-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)pyridine-3-carbonitrile
4-({4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}methyl)-5-(hydroxymethyl)-2-methylpyridin-3-ol