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1-[(4-chloro-3-fluorophenyl)methyl]-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
2-(2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetamido)-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
4-[4-(oxolane-2-carbonyl)piperazin-1-yl]quinazoline
2-chloro-4-{2-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}benzamide
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-4-amine
(2S)-2-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]formamido}-3-phenylpropanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-4-oxo-N-[phenyl(pyridin-4-yl)methyl]-2-propyl-1,4-dihydropyridine-3-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}aniline
4-[({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]-1-ethylpyrrolidin-2-one
3-(2-cyclopentylethyl)-N,N-diethyl-5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
dimethyl({2-[(oxolan-2-ylmethyl)({[2-(piperidin-1-yl)pyrimidin-5-yl]methyl})amino]ethyl})amine
5-(propan-2-yl)-N-[2-(pyridin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2-(6-methoxynaphthalen-2-yl)morpholine
methyl 4-[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]piperazine-1-carboxylate
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
N-(3-methylphenyl)-3-(1-phenylmethanesulfonylpiperidin-4-yl)propanamide
3-(furan-2-yl)-1-{4-[2-(3-methoxyphenyl)-1-[methyl(pyridin-2-ylmethyl)amino]ethyl]piperidin-1-yl}propan-1-one
1-(4-chlorophenyl)-N-({1-[3-(methylsulfanyl)propyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
1-{3-[(3-fluorophenyl)methyl]-1,2-oxazole-5-carbonyl}-3-(4-methoxyphenoxymethyl)piperidine
2-hydroxy-N-[(3R,4S)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-{2-[2-benzyl-5-oxo-4-(2-phenylphenyl)piperazin-1-yl]ethyl}acetamide
1-[6-(2-chloro-5-methylphenyl)pyridin-2-yl]ethan-1-ol
7-fluoro-N,N-dimethyl-2-[1-(3-methylpyridin-4-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]-2-oxo-1-phenylpyrrolidine-3-carboxamide
(2S,3R)-3-hydroxy-2-({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)butanamide
N-({5-[(3-hydroxy-4-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
methyl 2-(benzylsulfamoyl)-6-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}-N-phenylpiperidine-1-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
5-{[2-(2-hydroxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
3-[2-(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidin-1-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
1-[(3-methoxyphenyl)methyl]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
2-[4-(cyclopropylmethyl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
(1S,4S)-2-{[2-(1H-imidazol-2-yl)phenyl]methyl}-2-azabicyclo[2.2.1]heptane
3-(2-fluorophenyl)-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}propan-1-one
3-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
3,4-dimethyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N,N-dimethyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(quinoline-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1-ethyl-3-(2-methylpropyl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2-(morpholin-4-yl)propanamide
3-{[(1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
(3S,5R)-1-(2-chlorobenzoyl)-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
1-(5-chloro-2-methylphenyl)-4-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
[4-(1-benzyl-1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl](2-chloro-6-fluorophenyl)methanol
1-{1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carbonyl}piperidine-3-carboxamide