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1-benzyl-N5-cyclopropyl-N3-[(3-methoxyphenyl)methyl]-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[(3-chloro-1-benzothiophen-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(morpholin-4-yl)benzamide
propan-2-yl (4aS,7aR)-6,6-dioxo-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
1-[(2S)-2-[4-(cyclopropylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]pyrrolidin-1-yl]ethan-1-one
(1S,5R)-6-[(2-chloro-6-fluorophenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(pyridin-3-ylformamido)ethyl]piperidine-3-carboxamide
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(pyrimidin-2-yl)piperazin-1-yl]propan-1-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-6-(morpholin-4-yl)pyrimidin-4-amine
7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(2S,4S)-1-benzyl-4-{[(2,4-dimethoxyphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
ethyl 2-amino-3-cyano-4-(2-methoxypyrimidin-5-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-6-carboxylate
5-[4-(1-methyl-1H-pyrazol-4-yl)phenyl]-1,3,4-thiadiazol-2-amine
methyl 3-[(4-methoxy-2,5-dimethylphenyl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[2-(pyridin-3-yloxy)propyl]amine
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
3-(4-methyl-1H-pyrazol-1-yl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
8-methoxy-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
7-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(pyrrolidine-1-carbonyl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperazine
methyl 3-acetamido-5-{[4-(4-methoxyphenyl)butan-2-yl]amino}-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2-methoxy-5-methylphenyl)-2-({1-methyl-1H-pyrazolo[1,5-a]imidazol-7-yl}formamido)acetamide
2-(2-phenyl-1H-imidazol-1-yl)-N-[2-(pyridin-4-yl)ethyl]acetamide
4-{4-[(3S)-3-(3-methoxyphenyl)piperidin-1-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}pyridine
N-[2-(methylsulfanyl)ethyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
3,5-dimethyl-2-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1H-indole
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}propan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-(2-{[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
N-{3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-5-(aminomethyl)phenyl}pyridine-2-carboxamide
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-(furan-2-ylmethyl)urea
1-(furan-2-ylmethyl)-N-[2-(4-hydroxyphenyl)ethyl]piperidine-3-carboxamide
methyl (2S,4S)-4-(furan-2-amido)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
4-[1-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)piperidin-3-yl]benzoic acid
N-[(1-methylpiperidin-4-yl)methyl]-2-(morpholin-4-yl)-N-(2-phenylethyl)-2-(pyridin-3-yl)acetamide
N-[(2,3-difluoro-4-methylphenyl)methyl]-N-(pyridin-4-ylmethyl)cyclopropanamine
5-fluoro-2-[1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
8-[(2-chloro-4-fluorophenyl)methyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
(2S,4R)-N,N-diethyl-4-[2-(3-fluoro-4-hydroxyphenyl)acetamido]-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
2,6-dimethoxy-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
1-(furan-3-carbonyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
3-[(methylsulfanyl)methyl]-5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazole
3-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-4-methoxyphenol
2-amino-N-{2-[benzyl(methyl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl}-2-methylpropanamide