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3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
N-(2-methoxy-2-methylpropyl)-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
1'-(2-oxo-1,2-dihydroquinoline-3-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(3R,5R)-1-[(3,4-dimethoxyphenyl)methyl]-N-(2-methylpropyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
2-cyclopropanecarbonyl-8-[(furan-2-ylmethyl)carbamoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,5R)-6-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
8-{2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
6,7-dimethoxy-4-methyl-2-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}quinoline
2-benzyl-9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1-methylpiperidin-4-amine
benzyl(cyclopropylmethyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
[4-(3-phenylpropyl)-1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-4-yl]methanol
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(pyridin-4-yl)acetamide
{3-[(3-chlorophenyl)methyl]-1-(pyridin-2-ylmethyl)piperidin-3-yl}methanol
ethyl 1-{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}piperidine-4-carboxylate
1-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]urea
7-(5-chloropyridin-2-yl)-4-(2-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6,8-dimethyl-2-{[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}quinolin-4-ol
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-2-[(3S)-3-hydroxypyrrolidin-1-yl]-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
2-(4-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
3-chloro-4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}pyridine
2-(2,3-dimethoxyphenyl)-5-(pyrrolidin-1-ylmethyl)pyridine
1-(carbamoylmethyl)-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
2-[({[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}amino)methyl]-6-methyl-3,4-dihydropyrimidin-4-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
3-[2-(4-fluorophenyl)ethyl]-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
N-[(5-chloro-1H-indol-2-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
N-({1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-3-methylbut-2-enamide
2-{1-[(2-fluorophenyl)methyl]-4-[(2-methyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}cyclobutanecarboxamide
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-methyl-1,4-diazepan-5-one
5-methyl-3-[3-(pyridin-4-yl)azetidine-1-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-(2,5-dimethylphenyl)urea
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl][(1-propyl-1H-imidazol-2-yl)methyl]amine
4-ethyl-3-{1-[2-(4-hydroxyphenyl)acetyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-benzyl-N-[(3-methoxyphenyl)methyl]-N-methyl-1,3-benzoxazole-5-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-1H-indole-6-carboxamide
ethyl 5-{[2-(1-cyclopentyl-3-oxopiperazin-2-yl)acetamido]methyl}furan-2-carboxylate
N-cyclopropyl-4-methoxy-2-({1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-yl}oxy)benzamide
1-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(1H-1,2,3,4-tetrazol-5-yl)piperidine
1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(5-chlorothiophene-2-carbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]piperidin-2-one
4-(3-{3-[3-(2-methylpyridin-4-yl)phenyl]-1H-pyrazol-1-yl}propyl)morpholine
1-propyl-3-(thiomorpholine-4-carbonyl)-N-[(3,4,5-trimethoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(4-fluorophenyl)-N-{2-[7-(naphthalen-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
2-methoxy-N-[1-methyl-2-(pyridin-4-yl)-7-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1H-1,3-benzodiazol-5-yl]acetamide