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3-{3-[({[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}amino)methyl]-1H-indol-1-yl}propanamide
2-[5-(2-ethoxyethyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl]pyridine
{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-cyclopropyl-8-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(1-methyl-1H-pyrazole-3-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
6-[3-(prop-2-en-1-yloxy)benzoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-1-(4-phenylazepan-1-yl)propan-1-one
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-3-carboxamide
2-(5-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
2-[({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(propan-2-yl)amino]ethan-1-ol
3-[2-(2-hydroxyethoxy)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
methyl 6-[1-(4-methoxyphenyl)propan-2-yl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(5S,9aS,9bS)-5-(1,3-dimethyl-1H-pyrazol-4-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[1-methyl-5-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
7-(6-aminopyridine-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(1H-indol-1-yl)ethyl]-N,2-dimethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(2-{3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(3,6-dimethylpyrazin-2-yl)-N-methylpiperidin-3-amine
5-{[2-(diethylamino)ethyl](ethyl)amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidine
ethyl 4-(2-phenoxyethyl)-1-(thiophen-2-ylmethyl)piperidine-4-carboxylate
3-(3-fluorophenyl)-5-(thiophen-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-{2-[1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}acetamide
2-(4-methoxyphenoxy)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
(1S,5R)-3-(2,1,3-benzoxadiazol-4-ylmethyl)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(furan-3-carbonyl)-N-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-3-(2-fluorophenyl)pyrrolidine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
N-[(1S)-1-(1-cyclohexyl-3-phenyl-1H-1,2,4-triazol-5-yl)-2-(1H-imidazol-4-yl)ethyl]acetamide
2-methyl-6-{1-[2-(1H-1,2,4-triazol-5-yl)benzoyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
8-[4-(1H-pyrazol-3-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
2-[6-(benzyloxy)pyridin-3-yl]-3-(pyrrolidine-1-carbonyl)pyridine
N-{1-[4-(dimethylamino)phenyl]propan-2-yl}-2-(1-methylpiperidin-4-yl)acetamide
6-ethoxy-3-[(3-ethylpiperazin-1-yl)methyl]-1,2-dihydroquinolin-2-one
3-(azepane-1-sulfonyl)-5-(3,4-dimethoxyphenyl)benzoic acid
(3S,4R)-4-(3-fluorophenyl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidine-3-carboxylic acid
2-{4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-1,4-diazepan-1-yl}-1,3-benzoxazole
1-(1,4-dithiepan-6-yl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
4-[(3-fluorophenyl)methyl]-1-(2-methoxy-2-phenylacetyl)-1,4-diazepan-5-one
1-[(1S,5R)-6-[3-(4-hydroxyphenyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(3S,4S)-4-(piperidin-1-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidin-3-ol
2-{4-[(3,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-(dimethylamino)propan-2-ol
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-[(2-methoxyphenyl)methyl]-2-methyl-N-(prop-2-en-1-yl)-1,3-thiazole-4-carboxamide
(2R,6R)-4-(2-cyclopropylacetyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(furan-3-carbonyl)-4-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-1,4-diazepan-6-ol
1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-4-(3-methoxybenzoyl)piperazine
(3R,4R)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-(4-phenylbenzoyl)piperidine