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1-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N'-(2,4-dimethylphenyl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]propanediamide
1-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
8-(4-fluorobenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-butyl-4-(2-methoxyquinoline-4-carbonyl)-1-methylpiperazin-2-one
3-methyl-N-({1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-3-yl}methyl)but-2-enamide
1-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
2-[(3-methoxyphenyl)sulfanyl]-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
7-(3,6-dimethylpyrazin-2-yl)-4-(1,3-thiazol-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 2-[methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})amino]acetate
7-(2-methoxyacetamido)-1-methyl-2-phenyl-N-[1-(thiophen-3-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
5-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]propan-1-one
2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4-(pyrrolidin-1-yl)benzamide
1-(4-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-4-oxobutyl)pyrrolidin-2-one
3-methyl-1-({4-[3-(morpholin-4-yl)propoxy]phenyl}methyl)piperidin-3-ol
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-3-(naphthalen-1-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-3-(2H-1,3-benzodioxol-5-yl)propan-1-one
N2,N2-dimethyl-6-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidine-2,4-diamine
1-[(4-chlorophenyl)methyl]-N-(oxolan-2-ylmethyl)-N-propyl-1H-1,2,3-triazole-4-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(2-methylphenyl)piperidin-1-yl]ethan-1-one
3-ethyl-8-[(3S)-3-hydroxy-3-phenylpropyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]-1-methylpyrrolidin-2-one
2-{4-[3-(2-methyl-1H-indol-1-yl)propanoyl]morpholin-3-yl}acetic acid
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-(2-oxopyrrolidin-1-yl)acetamide
1-({methyl[1-(1,3-thiazol-5-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
N4,N4,5-trimethyl-N2-[1-(pyrazin-2-yl)propan-2-yl]pyrimidine-2,4-diamine
4-amino-2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]pyrimidine-5-carbonitrile
4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-(methylsulfanyl)-1,3-thiazole
3-{1-[1-(adamantan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
methyl (2S,4R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-[3-(4-methylphenyl)propanamido]pyrrolidine-2-carboxylate
4-{methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]carbamoyl}pyridin-1-ium-1-olate
(2S,4S)-1-benzyl-4-{[(3-ethoxy-4-methoxyphenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
6-[(3-fluorophenyl)methoxy]-4-(1-methyl-1H-pyrazole-5-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-benzotriazole-5-carboxamide
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazole
5-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyrazin-2-ol
(3R,4S)-4-(4-{2-methylthieno[3,2-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)oxolan-3-ol
[(3-{[1-(benzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-3-ylmethyl)amine
6-(3-fluorophenyl)-N-(2-methoxyethyl)-N-(propan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-phenyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
3-[2-(3-methoxyphenoxy)ethyl]-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2-methyl-4-(2-methylphenyl)piperazine
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(2-methylpropyl)amino]methyl}piperidin-2-one
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-benzyl-8-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
3-(1-{1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-1-ol