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N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N,8-dimethyl-3-{[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-{2-[(3-methoxypyrrolidin-1-yl)methyl]phenoxy}acetic acid
1-{1-[2-(3-fluorophenyl)acetyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-methylthiophene-2-carboxamide
1-(4-methylquinazolin-2-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
N-(1-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
2-[(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)methyl]benzonitrile
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-[(2,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-2-(1-methyl-3-oxopiperazin-2-yl)-N-(2-methylpropyl)acetamide
5-(azocane-1-carbonyl)-N-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
methyl 1-({4-[1-(pyridin-2-yl)piperidine-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
1-cyclopentyl-N-methyl-N-[(5-methyl-1H-indol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
6-[(2,6-difluorophenyl)methyl]-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-({3-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-3-ol
(2S,4S)-N-ethyl-4-[4-({methyl[(4-methylphenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-methyl-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-4-phenylbutane-1,4-dione
1-[(5-chlorofuran-2-yl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
3-[(2-fluoroethyl)sulfamoyl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
4-(4-acetamido-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)benzamide
N,N,4-trimethyl-3-({[(2-methylphenyl)methyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-cyclopropyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}-N-(1,3-thiazol-2-ylmethyl)acetamide
N-({7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
N-(3-hydroxyadamantan-1-yl)-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carboxamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
(3aR,6aR)-2-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
(1R,3S)-7-[(5-chlorothiophen-2-yl)methyl]-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
(1S,5R)-3-(pyridin-2-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)-4,6,7-trimethylquinazoline
2-methyl-5-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
methyl 2-{[(4-methylphenyl)methyl]sulfamoyl}-6-(1,2,5-thiadiazole-3-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(3-methoxyphenyl)-5-(oxan-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-{[4-(3-chlorophenyl)-5-({[(3,5-dimethoxyphenyl)methyl](methyl)amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
N-cyclopropyl-2-(methylamino)-N-{[4-(methylsulfanyl)phenyl]methyl}pyridine-4-carboxamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
1-(5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-4-methylpiperazine
5-(1-benzofuran-2-yl)-3-methyl-1H-1,2,4-triazole
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methoxypropanamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
3-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]thiophene-2-carboxamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine-4-carboxylate
dimethyl[(5-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]amine
N-[(1R,3R)-3-aminocyclopentyl]-4,5-dichlorothiophene-2-sulfonamide
6-fluoro-2-[({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)methyl]quinolin-4-ol
6-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
2-methyl-N-{2-[4-(4-methylphenoxy)piperidin-1-yl]-2-oxoethyl}propanamide
8-(1,3-benzothiazol-2-ylmethyl)-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione