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7-fluoro-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}quinazolin-4-amine
3-{2-[3-(ethoxycarbonyl)-3-[(4-fluorophenyl)methyl]piperidin-1-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate
(4-benzyl-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)methanol
2-(butylsulfanyl)-6-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}pyrimidin-4-amine
(1R,5R)-6-(2-methoxyethyl)-3-(4-methyl-2-phenylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-cyclohexyl-3-(cyclopropylmethyl)-N-[(3-methylpyridin-4-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-{2-[4-(dimethylamino)phenyl]ethyl}oxane-2-carboxamide
3-(3-chlorobenzoyl)-1-[(2,6-dimethoxyphenyl)methyl]piperidine
1-(5-methyl-1,2-oxazole-3-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
4-methyl-N-{[8-(pyridine-2-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
1-(quinoline-4-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[(3-fluorophenyl)methyl]-1-{imidazo[1,2-a]pyridine-2-carbonyl}-1,4-diazepan-5-one
(1H-indol-2-ylmethyl)({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N,N-bis(prop-2-en-1-yl)acetamide
{9-[(2-aminopyridin-3-yl)methyl]-3-benzyl-3,9-diazaspiro[5.5]undecan-1-yl}methanol
7-(2,6-dimethoxyphenyl)-4-[(4-fluorophenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1r,4r)-4-({5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)cyclohexan-1-ol
6-chloro-2-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methoxypyridine
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}urea
1-(4-{5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-1,4-diazepan-1-yl)ethan-1-one
1-(3-chlorophenyl)-4-[2-(1-ethylpiperidin-4-yl)acetyl]-5-methylpiperazin-2-one
2-(3-methoxypropyl)-9-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}acetamide
N-[3-(3-methylphenyl)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
2-(quinolin-3-yl)benzamide
4-[(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-2-methoxyphenol
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(furan-2-ylmethyl)acetamide
2-{1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}-1,3-benzoxazole
2-(2-{[(1R,2S)-2-phenylcyclopropyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-4-(4-fluorophenyl)butane-1,4-dione
1-(4-{[(cyclopropylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
2-methyl-6-[2-(naphthalen-1-ylmethyl)morpholine-4-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
2,2-bis(prop-2-en-1-yl)-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(4-fluorophenyl)methyl]-5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
N-(2-{1-[(2E)-3-phenylprop-2-en-1-yl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)acetamide
methyl 1-[(3R,5S)-5-[(1,3-dihydro-2-benzofuran-5-yl)carbamoyl]-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3,3-dimethyl-1-[(5-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
ethyl 4-(2-phenoxyethyl)-1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidine-4-carboxylate
3-(2-methoxyphenoxy)-1-(3,3,3-trifluoro-2-methylpropyl)azetidine
N-[(2,4-dimethoxyphenyl)methyl]-2-[2-(pyrrolidin-1-ylmethyl)-4-(thiophen-2-yl)phenoxy]acetamide
N-(1-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
2,6,6-trimethyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-1-propyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-methyl-N-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}oxan-4-amine
(3R,4R)-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-3,4-dimethylpyrrolidin-3-ol
3-(2-methoxyphenyl)-1-[3-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]propan-1-one
3-(2-amino-1,3-thiazol-4-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
2-(cyclopropylamino)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}acetamide