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[3-ethyl-1-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-3-yl]methanol
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(oxolan-3-ylmethyl)piperidine
2-[2-(methylsulfanyl)acetyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
5-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-(trifluoromethyl)-1H-1,3-benzodiazole
2-(1-ethylpiperidin-4-yl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]acetamide
2-ethyl-4-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)pyrimidine
1-ethyl-4-{[3-(1,2,3,6-tetrahydropyridine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperazine
2-ethyl-9-(2-methyl-1H-pyrrole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
N'1-methyl-N'1-[1-(3-phenylpropyl)piperidin-3-yl]cyclopropane-1,1-dicarboxamide
(2S,4S,5R)-4-[(1,3-dihydroxypropan-2-yl)carbamoyl]-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
5-{[cyclopropyl(3-methylpyridin-2-yl)methyl]carbamoyl}thiophene-2-carboxylic acid
7-methyl-3-[2-(piperazin-1-yl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
(2S,4R)-N-methyl-4-(4-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
4-{6-[4-(pyrrolidin-1-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
N-[(2R,3R)-1'-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
N-cyclopropyl-1-{1-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}piperidine-4-carboxamide
2-[4-(benzyloxy)butyl]-5-(dimethylamino)-2,3-dihydropyridazin-3-one
4-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
5-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
3-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-(2-methyl-1,3-benzothiazol-5-yl)urea
1-[(4-fluorophenyl)methyl]-4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
3-(2-methylpropyl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1,2-oxazole-5-carboxamide
N-[4-(1H-indol-2-yl)phenyl]-1-(pyrazine-2-carbonyl)piperidine-4-carboxamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-3-ol
1-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-methoxyethan-1-one
[(2,2-dimethyloxan-4-yl)methyl](methyl)[2-(1H-pyrazol-1-yl)ethyl]amine
[(4-ethyl-5-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)piperidine-3-carboxylate
N-[4-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenyl]acetamide
1-(2-cyclohexylethyl)-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
1-[(3-fluorophenyl)methyl]-5-[4-(2-hydroxyethyl)piperidine-1-carbonyl]piperidin-2-one
methyl 3-acetamido-5-{[(4-ethoxyphenyl)methyl]amino}-1-ethyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{1-benzyl-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-propyl-N-(pyridin-4-ylmethyl)acetamide
3-({[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}sulfamoyl)-N-phenylbenzamide
1-[4-(pyridin-2-ylmethoxy)phenyl]-3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
6-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(2-methylphenyl)acetyl]pyrrolidine-3-carboxylic acid
N-(2-{9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-oxoethyl)acetamide
(3S,4R)-4-(3-fluorophenyl)-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)pyrrolidine-3-carboxylic acid
1-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
7-(5-methylthiophen-2-yl)-4-(pyridazine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[5-(furan-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-(naphthalen-1-ylmethyl)acetamide