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1-(cyclopent-1-ene-1-carbonyl)-N-(3-fluorophenyl)piperidin-3-amine
1-(3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
1-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-ethyl-3-{[1-(9H-purin-6-yl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-methoxypropan-1-one
[5-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methyl)-4-phenyl-4H-1,2,4-triazol-3-yl]methanol
1-[4-(4-methoxyphenyl)piperazin-1-yl]-3-(3-methylpiperidin-1-yl)propan-1-one
2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[2-(pyridin-3-yl)ethyl]acetamide
2-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
1-[2-(4-benzyl-3-butyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetyl]piperidine-3-carbonitrile
5-(3-methylbut-2-en-1-yl)-1'-[(1-propyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
3-[(1,4-dimethylpiperazin-2-yl)methyl]-1-[4-(3-methylphenyl)phenyl]urea
1-[1-(oxan-4-yl)piperidine-4-carbonyl]-4-(pyridin-4-yl)piperazine
1-[(3-fluorophenyl)methyl]-4-[(6-methoxypyrimidin-4-yl)amino]pyrrolidin-2-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
ethyl 2-{2,7-diazaspiro[4.5]decan-7-yl}acetate
3-cyclopropyl-1-(2-ethylphenyl)-N-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazole-5-carboxamide
[(5-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}thiophen-3-yl)methyl]dimethylamine
7-(3-phenylpropyl)-2-[2-(pyridin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-1-methyl-1H-indole
1-[3-(1H-pyrazol-3-yl)phenyl]isoquinoline
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-4-oxo-4-phenylbutanamide
(3S,4S)-1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
(3S)-3-ethyl-4-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]morpholine
3-methyl-7-[(2E)-4-methylpent-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1,2,5-trimethyl-1H-pyrrole-3-carboxamide
[1-(1-hexylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanol
1-[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]-2-(2,3,6-trifluorophenyl)ethan-1-one
N-(furan-2-ylmethyl)-N,1-dimethyl-5-[(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-methyl-4-[(1-methyl-1H-imidazol-5-yl)methyl]-1-(2-methylpropyl)piperazin-2-one
2-ethoxy-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyridine-3-carboxamide
4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-4-(thiophen-2-yl)butan-1-one
N-cyclopropyl-3-acetamido-N-[(4-ethoxyphenyl)methyl]propanamide
3-[(4-chlorophenyl)methyl]-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
9-(4-hydroxy-3-methylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazine-1-carboxamide
3-({2-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[3-(oxolan-3-yl)-5-[(2,3,6-trifluorophenyl)methyl]-1H-1,2,4-triazol-1-yl]benzoic acid
4-(5-methoxypyridin-3-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
{1-[(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanamine
N-methyl-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-amine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
1-{7-[(2,4-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-methylpropan-1-one
2-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-(4-hydroxyphenyl)acetic acid
2-{5-cyclopropyl-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(thiophen-2-yl)pyrimidine
4-[(2S,4R)-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carbonyl]morpholine
N-[(2-fluorophenyl)methyl]-3-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-3-yl}propanamide