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{3-[(4-fluorophenyl)methyl]-1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl}methanol
1-methyl-2-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-2,5,7-trimethylquinoline
4-(1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)morpholine
6-(2-fluorophenyl)-N-[2-(3-methylpyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(2-chlorophenyl)methyl]-1-methyl-N-(prop-2-en-1-yl)-1H-pyrrole-2-carboxamide
1-(propan-2-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-4-carboxamide
1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridine-4-carboxamide
1-cyclopropyl-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
{1-[4-(4-{[(2,6-dimethoxyphenyl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
4-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
2-[4-(1H-indol-2-ylmethyl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}propanamide
4-[(1S,2R)-1-hydroxy-2-[2-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]propyl]phenol
[(2S,6S)-4-(2-propyl-1,3-thiazole-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(cyclohex-3-ene-1-carbonyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2-{2-[1-(3-chloro-2-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-2-(prop-2-en-1-ylsulfanyl)propanamide
(3S)-1-(8-methoxyquinolin-2-yl)pyrrolidin-3-ol
1-phenyl-4-[5-(2-phenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1H-pyrazole
2-methyl-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-1,4-diazepan-5-one
1-[(2-methoxyphenyl)methyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(4-ethylphenyl)methyl]methylamine
4-{6-amino-5-cyano-4-[3-(methoxycarbonyl)-1H-pyrazol-4-yl]pyridin-2-yl}benzoic acid
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[3-(prop-2-en-1-yloxy)phenyl]methyl}amine
N-(1-hydroxybutan-2-yl)-N'-(4-methylphenyl)-N-(pyridin-2-ylmethyl)propanediamide
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(2-methylphenyl)methyl]propanamide
1-{4-[4-(3-aminopyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}-3-methoxypropan-1-one
(1R,9aR)-1-[({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
1-[7-(1-benzothiophen-3-yl)-9-ethoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
[(3R,4R)-1-(1-phenylcyclopentanecarbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
[4-benzyl-1-(1-ethylpiperidin-3-yl)piperidin-4-yl]methanol
N-{[7-(5-propyl-1,2-oxazole-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(trifluoromethyl)benzamide
1-(1-cyclopentylpiperidin-4-yl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[4-(furan-2-yl)phenyl]-1-(oxane-4-carbonyl)piperidine-3-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
1-cyclopentanecarbonyl-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]piperidine
N-cyclopropyl-3-{1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidin-4-yl}propanamide
N-[(5-chloro-1H-indol-2-yl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-[(4-methoxyphenyl)amino]-2-methylpropan-1-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
8-{2-[2-(trifluoromethyl)phenyl]acetyl}-2,8-diazaspiro[4.5]decan-3-one
2-cyclohexyl-N-{imidazo[1,2-a]pyrazin-3-ylmethyl}acetamide
1-(propan-2-yl)-4-{2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}pyrrolidin-2-one
2-phenyl-N-(propan-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
(3aR,7aS)-2-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole