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1-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
3-ethyl-8-[(4-methylphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
4-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-pyrazole
3-(1-ethyl-1H-imidazol-2-yl)-1-[4-(2-fluorophenyl)benzoyl]piperidine
3-(4-acetylphenyl)-1-(oxolan-2-ylmethyl)-1-(2-phenoxyethyl)urea
2-[(3R,4S)-3-(3-methoxy-4-methylbenzamido)-4-(propan-2-yl)pyrrolidin-1-yl]acetic acid
N-[2-(1H-indol-3-yl)ethyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
8-(oxolan-2-ylmethyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(2,3-difluorophenyl)methyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(pyridin-3-ylmethyl)piperazine
N-[(2S,4R,6S)-2-ethyl-6-[2-(morpholin-4-yl)quinolin-3-yl]oxan-4-yl]acetamide
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
N-(3,4-difluorophenyl)-6-{2-[4-(methylsulfanyl)phenyl]acetyl}-6-azaspiro[2.5]octane-1-carboxamide
3-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-propyl-1-benzofuran-2-carboxamide
1-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-1,3-dimethyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-methyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-methyl-N-[(5-methylpyrazin-2-yl)methyl]-3-phenylcycloprop-2-ene-1-carboxamide
(4aR,8aR)-2-[5-(methoxymethyl)furan-2-carbonyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
3-(3-chlorobenzoyl)-N-(2,6-dimethylphenyl)piperidine-1-carboxamide
N-{3-[2-butyl-4-(4-chlorophenyl)-5-oxopiperazin-1-yl]-3-oxopropyl}acetamide
1-[6-(3-tert-butyl-5-methylphenyl)pyridin-2-yl]ethan-1-ol
2-[(4-methoxyphenyl)methyl]-N-methyl-N-[3-(morpholin-4-yl)propyl]-1,3-benzoxazole-6-carboxamide
(3S,4S)-4-cyclopropyl-1-[3-(dimethylamino)benzoyl]pyrrolidine-3-carboxylic acid
3-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}pyridin-2-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-15-methyl-13-oxo-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
3-[2-(dimethylamino)ethyl]-5-[1-(2-methylbenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
4-(2-methoxyacetyl)-N-[4-(1H-pyrazol-5-yl)phenyl]-1,4-diazepane-1-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
methyl 3-[(3S,4R)-1-[(3,4-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
2-(3-fluorophenyl)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]azepane
5-ethyl-5-{1-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]piperidin-4-yl}-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-propyl-1,2,4-oxadiazol-3-yl)piperidine
8-(9H-fluoren-2-ylmethyl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}-3-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea
2-methyl-5-{[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]acetamide
5-(oxolan-2-yl)-3-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1,2,4-oxadiazole
5-ethyl-1'-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazole
4-hydroxy-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-cycloheptyl-6-oxo-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-3-carboxamide
N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)oxolane-3-carboxamide
2-[(4-methylphenyl)amino]-2-phenyl-N-[2-(pyridin-2-yl)ethyl]propanamide
(3R,4R)-3-cyclopropyl-1-(3,4-dihydro-2H-1,5-benzodioxepine-7-sulfonyl)-4-methylpyrrolidin-3-ol
5-(2,6-dimethylphenoxymethyl)-N-(2-phenylpropyl)-1,2-oxazole-3-carboxamide