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2,6-dimethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]imidazo[1,2-a]pyridine-3-carboxamide
5-{1-[1-(propan-2-yl)piperidine-4-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-amino-7-[2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(2-fluorophenoxy)ethyl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-(thiophen-2-ylmethyl)benzamide
4-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}thiomorpholine
(2S,4S)-N-(1-benzothiophen-2-ylmethyl)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-[(3-methoxyphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-phenylbenzamide
1-(4-cyclohexylpiperazin-1-yl)-2-[4-(4-fluorophenyl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]ethan-1-one
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,6,8-trimethylquinoline-4-carboxamide
3-[1-(carbamoylmethyl)-1H-imidazol-2-yl]-N-(2-phenylethyl)piperidine-1-carboxamide
2-phenyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})amino]propane-1,2-diol
{2-oxo-2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}urea
2-methyl-3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-N-(pyridin-3-ylmethyl)aniline
3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
2-benzyl-8-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2,8-diazaspiro[4.5]decan-3-one
N-(1H-imidazol-2-ylmethyl)-3-(3-methoxypyrrolidine-1-carbonyl)-N-methylbenzene-1-sulfonamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-phenylethan-1-one
5-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]-1H-1,2,4-triazol-3-amine
[(1-benzylpiperidin-4-yl)methyl][(2-ethylpyrimidin-5-yl)methyl]methylamine
N-[(2,3-dimethoxyphenyl)methyl]-1-(oxan-4-yl)piperidine-4-carboxamide
5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-3-chloro-1,2-dihydropyridin-2-one
2-(2-ethoxybenzoyl)-2,7-diazaspiro[4.5]decane
N2-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-N4-ethylpyrimidine-2,4-diamine
3-(5-methyl-1H-pyrazol-1-yl)-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)propanamide
N-methyl-2-[1-(quinolin-4-ylmethyl)piperidin-4-yl]acetamide
N5,N5-dimethyl-N6-[1-(3-methylpyridin-2-yl)propan-2-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-(3-phenylpropyl)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
3-[(2-fluoro-5-methoxyphenyl)methyl]-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-{3-methyl-5-[2-(2-oxopyrrolidin-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
3-(2-chlorophenyl)-1-(pyridin-4-ylmethyl)-6-[2-(thiophen-3-yl)acetyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[1-(thiophen-2-yl)ethyl]benzamide
2-methoxy-5-({methyl[1-(2-phenylethyl)piperidin-3-yl]amino}methyl)phenol
2-(3-methoxyphenoxymethyl)-N-(oxan-2-ylmethyl)-1,3-oxazole-4-carboxamide
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)benzamide
2-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pyridine-3-carboxamide
5-[4-(morpholin-4-yl)piperidin-1-yl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-({1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}oxy)pyridine
2-(3-propyl-1,2-oxazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
1-methyl-1'-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
2-{[(3-ethoxyphenyl)methyl](2-phenylethyl)amino}ethan-1-ol
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-[(cyclohexylmethyl)amino]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
3-[(dimethylamino)methyl]-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-ol
N-[1-(cyclohexylcarbamoyl)piperidin-4-yl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperidin-2-yl)pyridine
1-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
5-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]-1H-1,3-benzodiazole