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[(3R,4R)-1-(4-methylpyrimidine-5-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-{1-[3-(furan-2-yl)benzoyl]piperidin-3-yl}benzoic acid
2-{4-[(6-methoxy-2H-chromen-3-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]thiomorpholine-4-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-(prop-2-en-1-yl)pyrrolidin-2-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-ethyl-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(2,3-difluorophenyl)methyl]-3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}[(4-methoxyphenyl)methyl]amine
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(furan-2-yl)phenyl]piperidine-3-carboxamide
N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-4-sulfamoylbenzamide
2-(3-chloro-4-hydroxyphenyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
2-{4-[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-1-yl}-N,N-dimethylacetamide
N-{[1-(methoxymethyl)cyclopentyl]methyl}-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
[(2S,4R)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(dimethylamino)pyrrolidin-2-yl]methanol
1-[2-(1-benzothiophen-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-ethyl-N-(2-methylprop-2-en-1-yl)piperidine-4-carboxamide
1-[(3-methoxyphenyl)methyl]-N-[3-(4-methylphenyl)propyl]-6-oxopiperidine-3-carboxamide
5-benzenesulfonamido-N,1-diethyl-2-methyl-N-(pyridin-4-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(naphthalen-1-yl)urea
1-[1'-(1-methyl-1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
8-fluoro-2-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1,4-dihydroquinolin-4-one
3-[(4-fluorophenyl)methyl]-5-methyl-5-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-(methoxymethyl)piperidine
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}pyridine-4-carboxamide
7-(3-chlorophenyl)-4-[(4-methoxy-3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-ethyl-1-[3-(5-methylfuran-2-yl)benzoyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
5-[1-(3-phenoxypropanoyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
3-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]-3-(2-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N,1-dimethyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1R,7S)-3-cycloheptyl-N-methyl-4-oxo-N-(thian-4-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
ethyl 1-[3-(dimethylcarbamoyl)propanoyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
(1H-indol-2-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
3-{[3-oxo-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzonitrile
2-[5,6-dimethyl-4-(1,2,3,6-tetrahydropyridin-1-yl)thieno[2,3-d]pyrimidin-2-yl]ethan-1-amine
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-(oxan-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-(cyclobutylmethyl)-2-[1-cyclopentyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)acetamide
{4-[(8-methoxy-2H-chromen-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
(5-{[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amino]methyl}furan-2-yl)methanol
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyridine-3-carboxamide
2-(4-hydroxyphenyl)-1-[3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
4,6-dimethyl-2-[({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-3-carbonitrile
(1S,5R)-3-[3-(1H-imidazol-2-yl)benzoyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}piperidine-3-carboxylic acid
3-cyano-N-[2-(pyridin-3-yloxy)propyl]benzamide
(2S)-3-methyl-2-(3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamido)butanamide
2-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-5-methoxyphenol
2-[4-(4-methoxyphenyl)-3-oxopiperazin-1-yl]-N,N-dimethylpropanamide
3-(2-methoxyethyl)-1-(2-phenylethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 1-ethyl-5-{[1-(2-fluorophenyl)propan-2-yl]amino}-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate