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{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
N-benzyl-N-methyl-1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-3-amine
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-{[(2,5-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-({[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}methyl)-1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
3-(2,3-dimethoxyphenyl)pyrazolo[1,5-a]pyridine
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-2-(2-methylphenyl)acetamide
1-methyl-5-(oxan-2-ylmethyl)-1H-indole
4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]phenol
4-{3-[4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]propyl}-1,3-thiazol-2-amine
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]propan-1-one
3-(2-methyl-5-oxo-1,4-diazepan-1-yl)-N-(4-methylphenyl)-3-oxopropanamide
4-cyclobutyl-6-methyl-N-[3-(4-methylpiperazin-1-yl)butyl]pyrimidin-2-amine
ethyl 5-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-[(4-methoxy-3-methylphenyl)methyl]-3-{2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
4-(4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)-1,4-diazepane-1-carbaldehyde
(3S,4R)-N,N-dimethyl-1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-4-(propan-2-yl)pyrrolidin-3-amine
N-cyclopropyl-4-methoxy-2-{[1-(3-phenylpropyl)piperidin-4-yl]oxy}benzamide
4-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}thiophene-2-sulfonamide
3,4,7-trimethyl-N-(pyrrolidin-2-ylmethyl)-1H-indole-2-carboxamide
2-(2-methoxy-5-methylphenyl)-2-{[(1-methyl-1H-imidazol-2-yl)methyl](propyl)amino}acetic acid
4-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-4-yl}thiomorpholine
3-ethyl-1-{[1-(naphthalen-1-ylmethyl)pyrrolidin-3-yl]methyl}urea
N-benzyl-N-methyl-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-amine
2-[(4-chlorophenyl)methyl]-8-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]-2-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)acetamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-[2-(2-ethoxyethoxy)phenyl]urea
methyl 2-{5-[1-(4,5,6,7-tetrahydro-1,3-benzothiazole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetate
1-[(1S)-1-[1-(4-chloro-2-methylphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl]-1H-1,2,3,4-tetrazole
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-[3-(trifluoromethyl)phenyl]acetamide
2-[2-(2-ethylmorpholin-4-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
5-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-2-methoxyphenol
8-[(3-methoxyphenyl)methyl]-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-ethyl-1H-pyrazol-5-yl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
1-[2-(4-chlorophenyl)ethyl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propanoic acid
3-(1-{[1-(2-hydroxyethyl)piperidin-3-yl]methyl}-4-phenyl-1H-imidazol-5-yl)phenol
4-[4-({[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amino}methyl)phenyl]but-3-yn-1-ol
3-{2-oxo-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
2,2-dimethyl-N-[1-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]propanamide
2-[(quinolin-8-yloxy)methyl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1,3-oxazole-4-carboxamide
4-[4-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)phenyl]-2-methylbut-3-yn-2-ol
3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-[2-(3-methylphenyl)ethyl]benzamide
7-methyl-2-{2-[(2-methylphenyl)sulfanyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
4-(1H-imidazol-1-yl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidine-4-carboxylic acid
4-{4-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(4-methoxyphenyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]propan-1-one