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ethyl 4-{2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetyl}piperazine-1-carboxylate
(5S)-5-{[benzyl({[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
1-cyclopropyl-N-methyl-5-oxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}pyrrolidine-3-carboxamide
3-{3-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}amino)methyl]-1H-indol-1-yl}propanamide
N-[(2-ethoxyphenyl)methyl]-1,3-dimethyl-2,6-dioxo-N-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[2-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)cyclohexanecarboxamide
(1-benzothiophen-2-ylmethyl)({[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})methylamine
2-acetyl-8-(4-methyl-1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-(2,3-dimethylphenyl)-4-phenyl-1-[2-(1H-pyrazol-4-yl)ethyl]-1H-imidazole
(3S,4S)-3-hydroxy-4-(2-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H-imidazol-1-yl)-1λ6-thiolane-1,1-dione
(1s,4s)-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-amido]cyclohexane-1-carboxylic acid
ethyl 3-[(2-methylphenyl)methyl]-1-(pyridine-4-carbonyl)piperidine-3-carboxylate
N-(1-benzylpyrrolidin-3-yl)-3-{1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidin-4-yl}propanamide
2-{[4-(1-phenylethyl)-5-(pyridin-3-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
8-[2-(1H-imidazol-4-yl)ethyl]-N,N-dimethyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
1-{6-[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]pyridin-2-yl}ethan-1-ol
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-3-(4-methoxyphenoxymethyl)piperidine
1-(2-cyclohexylethyl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-{[2-(3-methyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]methyl}pyridine
4-{3-[(propylamino)methyl]phenyl}benzamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[2-(4-fluorophenyl)piperidin-1-yl]-3-methoxypropan-1-one
2-[(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
9-(6-methylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-chloro-2-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}quinoline
6-{1-[(1-ethyl-1H-indol-5-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
2-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}acetamide
2-methyl-4-{4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
2-butyl-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-2,5-dihydro-1H-pyrrole
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-(3-ethoxypropyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
N,3,6-trimethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-benzofuran-2-carboxamide
N-butyl-2-methyl-N-(thiophen-3-ylmethyl)imidazo[1,2-a]pyrimidine-3-carboxamide
4-{2-[2-(2,4-dimethoxyphenyl)-1H-imidazol-1-yl]ethyl}-3,5-dimethyl-1H-pyrazole
N-(1-ethyl-5-methyl-1H-pyrazol-3-yl)-4-{[4-(propan-2-yl)piperazin-1-yl]methyl}benzamide
1-(4,7-dimethylquinazolin-2-yl)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
1-cyclopentyl-6-oxo-N-(pyridin-3-yl)piperidine-3-carboxamide
2-(pyridin-4-yl)-5-[4-(thian-4-yl)piperazine-1-carbonyl]pyrimidine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(6-methylpyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 3-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-(6-methyl-2-phenylpyrimidin-4-yl)pyrrolidin-3-yl]methyl}piperidin-4-ol
1-(2,6-difluorobenzenesulfonyl)-N-(3,4-difluorophenyl)piperidin-3-amine
N-[5-(4-methylpiperidine-1-carbonyl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]furan-2-carboxamide
N-(1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
2-(4-cyclohexylpiperazin-1-yl)-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
N-methyl-N-{[2-(4H-1,2,4-triazol-4-yl)phenyl]methyl}cyclohexanamine
ethyl 2-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetate