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8-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2,8-diazaspiro[4.5]decan-3-one
2-(pyridin-4-ylmethyl)-9-[2-(pyrrolidin-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-amino-4-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
9-hydroxy-N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1-benzothiophene-2-carboxamide
1-(1-acetylpiperidin-4-yl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(2-phenylpropyl)-1H-pyrazole-3-carboxamide
5-(4-methyl-2-phenylpiperazine-1-carbonyl)-2-(pyridin-3-yl)pyrimidine
N-[(2R,3R)-1'-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
1-cyclohexyl-4-(3-fluorobenzoyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-(2-methoxyethyl)-3-(3-methoxyphenyl)-3-(2-oxo-2-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}ethyl)pyrrolidine-2,5-dione
N-(2H-1,3-benzodioxol-5-yl)-5-[2-(pyridin-3-yl)-1H-imidazol-1-yl]furan-2-carboxamide
(4aS,7aR)-1-(1,2,4-oxadiazol-3-ylmethyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-4-methyl-1-(5-methylpyrazine-2-carbonyl)piperidine-3,4-diol
4-amino-2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pyrimidine-5-carbonitrile
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
[(2S)-1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
(2S,4S)-N-ethyl-1-(3-methoxypropanoyl)-4-(5-methylthiophene-2-amido)pyrrolidine-2-carboxamide
N,N,6-trimethyl-2-[2-(phenoxymethyl)pyrimidin-5-yl]quinoline-4-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-(4-fluorophenyl)-1-(4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-[(3R,5S)-1-(furan-3-ylmethyl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-({7-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-benzyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-sulfonamide
N-[4-(2-fluorophenoxy)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
2-fluoro-5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
1-(1H-imidazol-4-ylmethyl)-4-(1H-indole-6-carbonyl)-1,4-diazepan-6-ol
2-cyclopropyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}acetamide
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperazin-2-yl}ethan-1-ol
N-(2-hydroxyethyl)-5-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-4-[4-(4-methylphenoxy)piperidine-1-carbonyl]-1,3-thiazol-2-amine
(3aS,6aS)-2-(2-amino-6-methylpyrimidin-4-yl)-5-[2-(dimethylamino)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 2-hydroxy-5-({5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}methyl)benzoate
N-cyclopropyl-1-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
(2S)-2-(hydroxymethyl)-N-{4-[(2-phenylethyl)carbamoyl]phenyl}pyrrolidine-1-carboxamide
2-{2-[(1-phenoxypropan-2-yl)amino]ethyl}-1,2-dihydrophthalazin-1-one
5-(oxolan-2-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]thiophene-2-carboxamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-[(3S,4R)-3-cyclopropyl-4-acetamidopyrrolidin-1-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
3-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-2,5-dimethylpyrazine
ethyl 4-{[1-benzyl-3-cyclopropaneamido-2-(methoxycarbonyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]amino}piperidine-1-carboxylate
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethyl-1,2,3-thiadiazole-5-carboxamide
1'-[(2-aminopyridin-3-yl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-({1-[(3S,5S)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)pyridine-3-carboxamide
6-[(2-chloro-4,5-dimethoxyphenyl)methyl]-N-[2-(3-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol