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N-cyclopropyl-3-(1-propylpiperidin-4-yl)propanamide
N,N-dimethyl-2-[(1S,5R)-6-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
3-[(2S)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
2-{4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyridine
N-[(8-{[4-(benzyloxy)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[1-(2-ethyl-1H-imidazol-1-yl)propan-2-yl]amine
3-(furan-2-yl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
methyl 3-({[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)benzoate
N-{2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-(1H-imidazol-4-ylmethyl)piperidine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-(2-{[ethyl(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)ethan-1-one
N-[3-(4-{[3-(1H-1,3-benzodiazol-2-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-3-methylbutanamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[(3-methylpyridin-4-yl)methyl]pyrrolidine-2-carboxamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)acetamide
[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl][1-(2-fluorophenyl)propan-2-yl]amine
3-{2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-4-methylpyrimidine-5-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-oxo-2H-chromene-3-carboxamide
8-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-4-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1,4-diazepan-2-one
N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-(1-benzyl-1H-pyrazole-4-carbonyl)-4-phenylpiperidin-4-ol
7-ethyl-N-[2-(2-fluorophenyl)ethyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
3-[(3S,4R)-4-amino-3-methoxypiperidine-1-carbonyl]benzoic acid
5-propyl-4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
(3S,4R)-1-[2-(2,3-dimethoxyphenyl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
N-(cyclohexylmethyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
(3S)-1-[3-(pyridin-4-yl)propanoyl]piperidine-3-carboxylic acid
4-[4-(3-cyclopropyl-1-propyl-1H-1,2,4-triazol-5-yl)phenyl]morpholine
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-[3-(pyridin-4-yl)propyl]-1H-1,3-benzodiazole-7-carboxamide
2-methoxy-1-{3-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxymethyl]piperidin-1-yl}ethan-1-one
1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(2-phenylethyl)piperazine
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-3-(1-methylpiperidin-2-yl)propanamide
N-{7-[2-(hydroxymethyl)piperidine-1-carbonyl]-1-(2-phenylethyl)-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
methyl(thiophen-3-ylmethyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
1-(3-methylpyridin-2-yl)-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-N-(2-phenylethyl)piperidin-3-amine
1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-(1,3-dimethyl-1H-pyrazol-5-yl)-3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}benzamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-indole-3-carboxamide
N-(3-hydroxypropyl)-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-[(6-chloropyridin-3-yl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]acetic acid
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
1-(3-methoxyphenyl)-3-methyl-3-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)urea
N-[3-(ethylcarbamoyl)-5-({[3-(5-methylfuran-2-yl)butyl]amino}methyl)phenyl]pyridine-2-carboxamide
1-cyclopropyl-5-oxo-N-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrrolidine-3-carboxamide