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2-(dimethylamino)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(4-fluorophenyl)acetamide
1-[7-(1-benzothiophen-3-yl)-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
2-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]pyridine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-[(3-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
6-ethyl-2-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)quinoline-4-carboxamide
5-methyl-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1-propyl-1H-pyrazole-4-carboxamide
8-[(2,6-difluorophenyl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-(thiophene-2-carbonyl)piperidine
(2R,4S)-1-(2,3-dihydro-1-benzofuran-7-carbonyl)-4-hydroxypiperidine-2-carboxylic acid
1-[3-(aminomethyl)phenyl]-3-(2-ethyl-2,5-dihydroxypentyl)urea
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1,4-dithiepan-6-amine
1-(3-methylbutyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
3-[1-(1-methoxypropan-2-yl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-(2,5-dimethylfuran-3-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-4-methylpyrimidine-5-carboxamide
3-[4-(2,3-dihydro-1H-inden-2-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
5-[3-(azepan-1-yl)-3-oxopropyl]-5-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-2-one
6-[(3,5-dimethoxyphenyl)methoxy]-4-(oxane-4-carbonyl)-1-(propan-2-yl)-1,4-diazepan-2-one
5-(2-fluorophenyl)-N-[3-(morpholin-4-yl)propyl]-1,2,4-triazin-3-amine
N,N-diethyl-1-{[1-(1-propylpiperidin-4-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]benzene-1-sulfonamide
N-{1-[1-(1-aminocyclopropanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
1-[2-({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-2-one
2-chloro-N-(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-(2-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]amino}ethyl)acetamide
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)ethan-1-one
(3S,9aR)-3-[(benzyloxy)methyl]-8-(4-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(dimethylamino)ethyl]-3-(4-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
5-({[2-fluoro-5-(trifluoromethyl)phenyl]methyl}carbamoyl)-1H-imidazole-4-carboxylic acid
N-[(3S,4R)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-(3-fluorophenyl)-6-[(2-methyl-1H-indol-3-yl)methyl]-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-cyclopropyl-N-(furan-2-ylmethyl)-4-hydroxy-N-(thiophen-2-ylmethyl)pyrimidine-5-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-(2-methoxyphenyl)acetamide
1-[(1-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-3-yl)methyl]pyrrolidin-2-one
3-[1-(adamantan-2-yl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
1-{2-[(4aS,8aR)-1-(3-aminopropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
6-{1-[(3-methyl-1,2-benzoxazol-5-yl)methyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-5-propyl-1,3,4-oxadiazol-2-amine
N,N-diphenyl-4-(1H-1,2,3-triazole-5-carbonyl)piperazine-1-carboxamide
1-(3-benzylphenyl)-3-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-methylurea
{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}bis(prop-2-en-1-yl)amine
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
dimethyl[1-(1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)ethyl]amine
1-[(2-aminopyridin-3-yl)methyl]-4-[4-(methylamino)pyrimidin-2-yl]-1,4-diazepan-6-ol
N-[(3,5-dimethoxyphenyl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-[(2S)-1-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
3-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
7-(cyclopropylmethyl)-2-(2-methoxyacetyl)-2,7-diazaspiro[4.5]decan-6-one
2-methoxy-N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-phenylacetamide
4-[1-(2,4-dimethoxybenzoyl)piperidin-3-yl]-5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidine