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N-[(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
2-amino-6-(4-hydroxyphenyl)-4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]pyridine-3-carbonitrile
4-[3-(1H-pyrazol-3-yl)phenyl]isoquinoline
4-methoxy-N-(2-methoxyethyl)-2-({1-[1-(pyridin-2-yl)propan-2-yl]piperidin-4-yl}oxy)benzamide
N5-cyclopropyl-N6-[(2-methylphenyl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(4S,4aS,8aS)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-phenyl-decahydroquinolin-4-ol
2-ethyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]pyrimidine-5-carboxamide
1-{2-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]ethyl}-4-methyl-1H-1,2,3-triazole
1-(4-fluorophenyl)-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazine
{5-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]furan-2-yl}methanol
N-[3-(3-chlorophenyl)phenyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine-4-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxamide
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-[(3,4-dimethylphenyl)methyl]urea
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
8-(6-aminopyridine-3-carbonyl)-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
7-[(3,4-difluorophenyl)methyl]-2-(oxane-4-carbonyl)-2,7-diazaspiro[4.5]decane
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(1r,4r)-4-hydroxycyclohexyl]amino}methyl)piperidin-2-one
[(4-ethynylphenyl)methyl](furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amine
2-{[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-5-methoxyphenol
1-[2-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)-2-oxoethyl]-4-phenylpyrrolidin-2-one
4-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-3-methyl-1-propyl-1H-pyrazole
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}propan-1-one
N,N-dimethyl-5-{[8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}pyridin-2-amine
1-(5-chloropyridin-2-yl)-4-(2-methoxypyridine-4-carbonyl)piperazine
N4-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-6-methylpyrimidine-2,4-diamine
4-[5-(5-methylpyrazin-2-yl)-1-propyl-1H-1,2,4-triazol-3-yl]benzamide
1-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
N-[3-(1H-indol-2-yl)phenyl]-1-(2-methylfuran-3-carbonyl)piperidine-3-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidine-4-carboxamide
dimethyl({2-[(6-methylpyridazin-3-yl)oxy]phenyl}methyl)amine
2-(morpholin-3-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
N-(2-fluorophenyl)-5-{1H-pyrazolo[3,4-b]pyridin-1-yl}furan-2-carboxamide
2-[5-(furan-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]quinoxaline
methyl 8-(3-ethynylbenzoyl)-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
6-hydroxy-N-(5,7,8-trimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1,4-oxazepane-4-carboxamide
6-({[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
3-[4-(benzyloxy)piperidin-1-yl]-5-(2-methylphenyl)-1,2,4-triazine
1-methyl-4-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,4-diazepane
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-[2-(dimethylamino)ethyl]-4-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]pyrrolidin-2-one
6-methyl-3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-methyl-6-{1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperidin-4-yl}pyrimidin-4-ol
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
2-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2-dihydrophthalazin-1-one
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
N-{5H,6H,7H,8H,9H,10H-cyclohepta[b]indol-2-ylmethyl}-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
4-fluoro-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}benzamide
1-ethyl-N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[4-(5-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
4-[7-(4-cyanopyridin-2-yl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide