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1-[(3-fluorophenyl)methyl]-5-[4-(methoxymethyl)piperidine-1-carbonyl]piperidin-2-one
4-[3-(ethoxymethyl)-5-(5-methylpyrazin-2-yl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
1-ethyl-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1H-pyrazole-5-carboxamide
N-[1-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
1-(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}azetidin-3-yl)-2-methylpiperidine
1-[3-(1H-imidazol-2-yl)benzoyl]-4-[(methylsulfanyl)methyl]piperidine
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-2-methyl-1,3-benzothiazole-5-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-5-(3-fluorophenyl)-1,2,4-triazin-3-amine
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl][2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]methylamine
2-{4-[4-(2-ethoxyphenyl)piperazin-1-yl]pyrimidin-5-yl}acetic acid
{[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}[(1-propyl-1H-pyrazol-4-yl)methyl]amine
4-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}pyridin-2-amine
2-{[({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)amino]methyl}-6-methoxyphenol
N'-(2,5-dimethylphenyl)-N-[2-(1H-imidazol-4-yl)ethyl]propanediamide
methyl 1-[(3R,5S)-1-(3-phenylpropyl)-5-[(thiophen-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
9-(1-aminocyclopropanecarbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-(3-phenylpropyl)-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3R,4S)-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3,4-dimethylpiperidin-4-ol
3-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}pyridin-2-amine
5-{[3-(2-methylphenoxymethyl)piperidin-1-yl]methyl}pyrimidin-2-amine
N-{2-[(2R,3R)-2-hydroxy-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-oxoethyl}methanesulfonamide
1'-(2,3-dihydro-1H-inden-2-yl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3S,4S)-4-(dimethylamino)-1-{[2-(2-phenylethoxy)phenyl]methyl}pyrrolidin-3-ol
4-[3-(aminomethyl)phenyl]benzoic acid
dimethyl[(5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}furan-2-yl)methyl]amine
N-[(3S,4R)-1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-4-propylpyrrolidin-3-yl]methanesulfonamide
2-(3-chlorophenyl)-4-[4-(furan-2-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3,3-difluoro-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}propanamide
5-{[benzyl(methyl)amino]methyl}-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
5-methoxy-N,3-dimethyl-N-(quinolin-5-ylmethyl)-1H-indole-2-carboxamide
1-[4-(4-hydroxybutyl)piperazin-1-yl]-3-(2-methyl-1H-indol-1-yl)propan-1-one
4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
2,4-dichloro-6-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)phenol
N-[3-(cyclohexylcarbamoyl)-2-methylphenyl]-3-methylthiophene-2-carboxamide
3-hydroxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}pyridine-2-carboxamide
3-cyclopropaneamido-4-methyl-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]benzamide
(3S,4R)-1-(5-ethylthiophene-3-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-(cyclopropylmethyl)-9-[(2-fluoro-5-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-5-[methyl(thiophen-2-ylmethyl)amino]-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[3-(5-methylfuran-2-yl)butyl]-4-phenoxypiperidine-4-carboxylic acid
1-(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-4-(furan-2-carbonyl)piperazine
[(4-{2-[4-(2H-1,3-benzodioxole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](1-benzothiophen-2-ylmethyl)methylamine
4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-N-(1,3,4-thiadiazol-2-yl)benzamide
N-methyl-N-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}thian-4-amine
N-cyclopropyl-3-{5-[(2-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide