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4-methyl-3-[3-(1H-pyrazol-3-yl)phenyl]benzoic acid
2-(1-cyclohexyl-4-{[2-(difluoromethoxy)phenyl]methyl}piperazin-2-yl)ethan-1-ol
2-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-methylphenyl)-3-phenylpropanamide
3-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]pyridine
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(morpholin-4-yl)ethyl]piperidine-3,5-dicarboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
8-[4-(hydroxymethyl)phenyl]-2-methylquinolin-4-ol
ethyl 1-(2-oxo-2-phenylacetyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
1-(2-ethoxyethyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-(2-ethylphenyl)-3-[2-(propan-2-yloxy)acetamido]benzamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
6-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-1-benzofuran-2-carboxamide
5-(2-fluoro-5-methoxyphenyl)-4-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
dimethyl({1-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-4-yl]ethyl})amine
[(4-fluoro-3-methoxyphenyl)methyl][(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amine
3-methyl-3-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(2,4,5-trifluorophenyl)urea
4-(2-ethyl-3-oxopiperazin-1-yl)-4-oxo-N-(2,4,6-trimethylphenyl)butanamide
2-[1-(2,5-dimethylfuran-3-carbonyl)pyrrolidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-1-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}urea
3-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
2-ethyl-4-methyl-N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-1,3-oxazole-5-carboxamide
5-chloro-6-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpyrimidin-4-ol
2-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
N-(1-propyl-1H-1,2,3-triazol-4-yl)-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
methyl 3-{4-[2-(methylsulfanyl)acetyl]-2-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl}propanoate
N-(3,5-dimethoxyphenyl)-3-{1-[3-(methylsulfanyl)propyl]piperidin-3-yl}propanamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]amine
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole
2-[2-(dimethylamino)ethyl]-8-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(2-amino-1,3-thiazol-4-yl)-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)propanamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}propanamide
(4aS,8aS)-2-({3-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-decahydroisoquinolin-4a-ol
N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-[5-(1H-imidazol-2-ylmethyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
8-fluoro-2-(3-hydroxyazetidine-1-carbonyl)-1,4-dihydroquinolin-4-one
4-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidine-1-carbonyl]-N-methylpyridin-2-amine
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}oxolan-3-amine
3-(3,4-difluorophenyl)-1-[3-(3-methoxyphenoxy)azetidin-1-yl]propan-1-one
2-cyclopentyl-2-phenyl-1-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
(2E)-3-(4-chlorophenyl)-1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]prop-2-en-1-one
(3aR,6aR)-N-(2H-1,3-benzodioxol-5-ylmethyl)-2-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
dimethyl[(5-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]amine
6-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-5-methyl-N-(oxolan-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
1-methyl-4-{6-[(propan-2-yl)amino]pyrimidin-4-yl}piperazine-2-carboxylic acid
3-{4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
(2S,4S,5R)-1,2-dimethyl-4-[(oxan-4-ylmethyl)carbamoyl]-5-phenylpyrrolidine-2-carboxylic acid