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5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]pyridine-2,4-diol
(2R)-2-amino-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-3-methylbutanamide
2-phenyl-N-[1-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
3-[3-(dimethylamino)propyl]-8-(1-methoxypropan-2-yl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
10-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-methyl-6-(3-methyl-3-phenylpiperidine-1-carbonyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-5-phenyl-1,2,4-triazin-3-amine
1-(3-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)ethan-1-one
2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-N-(2-phenylethyl)acetamide
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
1-(3-{[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}propyl)piperidin-3-ol
4-{1-[1-(3-methoxypyrazin-2-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1,4-oxazepan-6-yl)methanol
1-cyclobutanecarbonyl-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
1-methyl-4-(2-methyl-1-benzofuran-7-carbonyl)-1,4,9-triazaspiro[5.5]undecane
{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}bis(prop-2-en-1-yl)amine
N-(1-propylcyclopropyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(3-methoxypropyl)-8-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-(1H-1,2,3-benzotriazol-4-yl)-2-[4-(3-hydroxybenzoyl)morpholin-3-yl]acetamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-(1-hydroxy-3-methylbutan-2-yl)-1,2-oxazole-3-carboxamide
3-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-1-[3-(1H-imidazol-1-yl)propyl]urea
N-[(3R,4S)-1-(6-methylpyridazin-3-yl)-4-propylpyrrolidin-3-yl]-2-(morpholin-4-yl)acetamide
N-benzyl-3-(1-methylpiperidin-2-yl)-N-(1,3-thiazol-2-ylmethyl)propanamide
4-cyano-N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
4-[(3-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}phenyl)methyl]morpholine
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]acetamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
4-({4-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]furan-2-yl}methyl)morpholine
N-[2-(3,5-dimethylphenoxy)ethyl]-N-methyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(4-fluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
ethyl 4-[(4-chlorophenyl)methyl]-1-cyclobutylpiperidine-4-carboxylate
2-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2-oxo-2-phenylacetyl)piperidine-3-carboxylate
3-(2-amino-4-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-6-methylpyrimidin-5-yl)propanoic acid
2-methoxy-1-[1'-(1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-methyl-N-(oxan-4-yl)-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[(8-methoxyquinolin-5-yl)methyl]-N,2-dimethyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
1-cyclopropyl-5-oxo-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrrolidine-3-carboxamide
2-methyl-N-(2-phenylethyl)-N-propyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-(dimethylamino)-2-(3-methylphenyl)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
N-[1-(3-propyl-1,2,4-oxadiazol-5-yl)ethyl]-4-(1H-pyrazol-4-yl)butanamide
1-(3-{[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
1-[4-(furan-2-yl)pyrimidin-2-yl]-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-methyl-2-[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]acetamide
4-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]-1-(oxan-4-yl)piperidine
[3-(2-phenoxyethyl)-1-(2-phenylethyl)piperidin-3-yl]methanol
(3S)-1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-N,N-dimethylpyrrolidin-3-amine
methyl (2S)-1-{[4-(2,3-dihydro-1H-inden-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}pyrrolidine-2-carboxylate