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N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-(4-methoxyphenoxy)-N-methyl-N-(prop-2-en-1-yl)benzamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(1H-pyrrol-1-yl)pentanamide
2-(5-{[3-(4-fluorophenoxymethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
4-cyclobutyl-N,6-dimethyl-N-[2-(pyridin-2-yl)ethyl]pyrimidin-2-amine
3-{5-[(4-methoxy-2,5-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2,6-dimethylpyridin-4-yl)piperazine
5-acetyl-N,2,4-trimethyl-N-(pyrazin-2-ylmethyl)-1H-pyrrole-3-carboxamide
7-(3-fluoro-2-methoxybenzoyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
methyl 3-(oxolane-2-amido)-1-(2-phenylethyl)-5-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{4-[(4-cyano-4-phenylpiperidin-1-yl)methyl]phenoxy}propanoic acid
2-ethyl-N-{2-[(trifluoromethyl)sulfanyl]ethyl}pyrimidine-5-carboxamide
(3S,5R)-1-(1-benzofuran-2-ylmethyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
(1R,5R)-6-(1H-imidazol-2-ylmethyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
(4aS,8aS)-2-(4-methylphthalazin-1-yl)-decahydro-2,7-naphthyridin-4a-ol
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
3-cyclopropyl-N-(2-methylpropyl)-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazole-5-carboxamide
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
1-cyclopropyl-N-[3-(1H-imidazol-1-yl)propyl]-5-oxo-N-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-methoxy-4-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]pyridine
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-(4-propanoylphenoxy)acetamide
ethyl 2-[9-(2-ethylbutanoyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetate
(5-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-2-ethoxyphenyl)methanol
1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(thiophen-2-yl)propan-1-one
3-(4-methyl-1,3-thiazol-5-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}propanamide
5,6-dimethoxy-2-[(1-methylpiperidin-2-yl)methyl]-1,2-dihydroisoquinolin-1-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-methyl-2-[5-methyl-2-(propan-2-yl)phenoxy]propan-1-one
{2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}dimethylamine
(2S,4S)-4-({[4-(benzyloxy)phenyl]methyl}amino)-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]acetamide
3-{2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2,7,8-trimethyl-4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}quinoline
N-(1-methyl-1H-indazol-5-yl)thiomorpholine-4-carboxamide
methyl 4-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-1H-pyrazole-3-carboxylate
methyl 2-(1-{1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidin-3-yl}-N-methylformamido)acetate
3,5-dichloro-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N,4-dimethylbenzamide
(3aS,6aS)-2-cyclohexyl-5-[3-(1H-imidazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-(1-methyl-1H-imidazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(furan-2-ylmethyl)(methyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
8-(2-ethylpyrimidine-5-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(2-aminoethyl)-4-(5-chloro-2-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{2-oxo-2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,3-oxazolidin-2-one
1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(1H-pyrazol-3-yl)pyridine-3-carboxamide
2-[4-(dimethylamino)phenyl]-1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]ethan-1-one
1-methyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-1H-pyrazole-5-carboxamide