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[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]diphenylmethanol
N-[2-(1H-imidazol-4-yl)ethyl]-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
4-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-2-phenylmorpholine
1-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
1-[(1R,5R)-6-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}(quinolin-8-ylmethyl)amine
4-[(2,5-dimethoxyphenyl)methyl]-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{2-[3-(phenoxymethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidin-2-one
1-methyl-3-{[1-(4-phenylphenyl)piperidin-4-yl]amino}pyrrolidin-2-one
3-[2-(3,4-difluorophenyl)acetyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-({4-[(3,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-N,N-diethylpiperidine-3-carboxamide
4-fluoro-N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)benzamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-fluoro-6-methoxybenzamide
8-[2-(2,4-difluorophenyl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)pyrazine
(1R,5S)-3-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-propyl-1,3-thiazole-4-carboxamide
1-(2-methoxyethyl)-4-{[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}pyrrolidin-2-one
2-hydroxy-4-(methylsulfanyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}butanamide
1-{[2-({[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}methyl)phenyl]methyl}pyrrolidin-2-one
N-[(3,4-dimethoxyphenyl)methyl]-4-(morpholin-4-yl)-N-(pyridin-2-ylmethyl)benzamide
3-(3-methoxyphenyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2-(1H-1,2,3,4-tetrazol-5-yl)acetamide
(3aS,6aR)-5-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-methyl-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[(2-fluorophenyl)formamido]-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}propanamide
(3aS,6aS)-2-(4-cyclobutyl-6-methylpyrimidin-2-yl)-5-cyclopentanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[6-(4-hydroxypiperidin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
N5-cyclopentyl-N6-[(dimethyl-1,3-thiazol-2-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}oxy)benzamide
1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
2-{4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}acetamide
N,N-dimethyl-2-{[(5-methyl-1,3-benzoxazol-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
methyl 3-chloro-4-{[4-(2-methylpyrimidin-4-yl)piperidine-1-carbonyl]amino}benzoate
2-(furan-2-ylmethyl)-9-[2-(methylsulfanyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2,5-dimethoxy-N-(pyridin-4-ylmethyl)benzamide
(2S,4S)-N,N-diethyl-4-(furan-2-amido)-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
1-[7-(hydroxymethyl)-9-methanesulfonyl-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
1-cyclopropyl-4-[({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]pyrrolidin-2-one
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(3-chlorophenyl)methyl]piperidine
(3S,4R)-4-methyl-1-(2,3,4,9-tetrahydro-1H-carbazole-8-carbonyl)piperidine-3,4-diol
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1-phenylcyclopropane-1-carboxamide
5-(3,3-diphenylpiperidine-1-carbonyl)pyridine-2,4-diol
5-methyl-5-(4-methylpent-3-en-1-yl)-1-[2-(pyrazin-2-yl)ethyl]piperidin-2-one
8-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-4-(2-methoxybenzoyl)piperazine