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1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
8-(benzenesulfonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{2-[(5-tert-butyl-1,3,4-oxadiazol-2-yl)amino]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
8-cyclopropanecarbonyl-2-(thiophene-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,5R)-6-(3-chloro-4-methoxybenzoyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)oxolane-3-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(9H-purin-6-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
dimethyl({5-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]furan-2-yl}methyl)amine
1-(2-methoxyethyl)-2-[3-methyl-1-(2-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-imidazole
2-(5-{1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
N-[2-(4-chlorophenyl)ethyl]-2-[3-(N-methylacetamido)pyrrolidin-1-yl]acetamide
(3S,4R)-4-(2-methoxyphenyl)-1-(propan-2-yl)pyrrolidine-3-carboxylic acid
11-(4-ethyl-5-methylthiophene-3-carbonyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
9-[(4-methoxypyridin-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)urea
ethyl 4-[(4-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
2-[1-({1-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
4-(3-chlorophenoxy)-1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidine
N-propyl-4-{[3-(pyridin-2-yl)propyl]sulfamoyl}benzamide
4-(methoxymethyl)-1-{[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidine
N-{2-[3-cyclopropyl-1-(2,3-dimethylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
2-(3-methoxyphenyl)-5-(3,3,4,4-tetrafluorobutyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl)amino}-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
2-[2-hydroxy-5-(1H-pyrrol-1-yl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
[3-(cyclopropylmethyl)-1-(5-methoxypyrimidin-2-yl)piperidin-3-yl]methanol
5-{[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-N,N-dimethylpyrimidin-2-amine
3-(4-phenylbenzoyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
4-(oxan-2-ylmethyl)-1-{thieno[3,2-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
3-ethyl-N1-(2-methyl-5-sulfamoylphenyl)piperidine-1,3-dicarboxamide
4-[(dimethylamino)methyl]-1-(5,6-dimethylpyrimidin-4-yl)azepan-4-ol
2-{[(1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
2-methyl-3-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-4,5,6,7-tetrahydro-1-benzofuran-4-one
1-[1-(furan-3-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
N-[(1S)-3-methyl-1-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]butyl]acetamide
[(2,6-dimethoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-ethyl-2-{[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,3-thiazole
2-(4-{[4-(cyclopentyloxy)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
2,6,8-trimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}quinoline-4-carboxamide
2-(5-chlorofuran-2-carbonyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(3-methylpyridin-4-yl)pyrrolidin-3-yl]methanol
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butane-1,2-dione
N-(1-benzothiophen-2-ylmethyl)-2-[2-(pyrrolidin-1-ylmethyl)-4-(thiophen-2-yl)phenoxy]acetamide
3-{2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-[4-(propan-2-yl)piperazin-1-yl]pyridine-3-carboxamide
3-({[1-(4-propylbenzoyl)piperidin-4-yl]oxy}methyl)pyridine
N-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]morpholine-4-carboxamide
(3S,4S)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-propylpyrrolidine-3-carboxylic acid