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N-[(4-fluorophenyl)methyl]-3-{1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}propanamide
N-[(1-{[4-(pyridin-2-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]methanesulfonamide
N,4-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-pyrrole-2-carboxamide
2-[(3S,4R)-3-cyclopropyl-4-[(pyrimidin-2-yl)amino]pyrrolidin-1-yl]ethan-1-ol
1-[4-(cyclobutylmethyl)-6-hydroxy-1,4-diazepan-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
7-(3-chlorophenyl)-4-(2-methylfuran-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]-3-methyl-1-propyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-5-phenyl-1,2-oxazole-3-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-(1-methanesulfonylpiperidin-4-yl)benzamide
N,2-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}oxane-2-carboxamide
N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-benzothiazole-6-carboxamide
(2R)-5-oxo-N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]pyrrolidine-2-carboxamide
N-(4-chloro-2-methylphenyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
1-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-5-phenyl-1H-pyrrole-2-carboxamide
2-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
1-(2-chlorophenyl)-5-methyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-2-one
N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-1,2,3,4-tetrahydronaphthalene-2-carboxamide
3-chloro-N-(2-methoxyethyl)-4-{[1-(thiophen-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
2-(cyclopropylmethyl)-7-(1-ethyl-3-methylpiperidine-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4aR,6R,8aS)-2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
4-[1-hydroxy-2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]phenol
N-[(3-methyl-1-benzofuran-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[cyclohexyl(methyl)amino]-3-{2-[({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amino)methyl]phenoxy}propan-2-ol
3-benzyl-1-(3-cyano-4,6-dimethylpyridin-2-yl)piperidine-3-carboxylic acid
5-(2-chlorophenyl)-4-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-3-yl]pyrimidine
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-amine
1-(5-fluoropyridin-2-yl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-N,N-diethylpiperidine-4-carboxamide
2-{5-[2-(methylamino)-1,3-thiazol-4-yl]-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl}acetic acid
2-{5-[2-(1-methylpiperidin-2-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-{pyrazolo[1,5-a]pyridin-7-yl}pyridin-2-ol
4-(hydroxymethyl)-1-(3-phenoxybenzoyl)azepan-4-ol
2-[5-(2H-1,3-benzodioxol-5-yl)-1H-indol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
1-[3-({3-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
1-{1-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
(1-{furo[3,2-c]pyridin-4-yl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
2-methyl-1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-1,4-diazepan-5-one
methyl 3-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}furan-3-carboxamide
6-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}pyrimidin-4-amine
2-(4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidin-1-yl)acetic acid
3-(1-methylpiperidin-2-yl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]propanamide
1-[6-hydroxy-4-(isoquinolin-1-yl)-1,4-diazepan-1-yl]ethan-1-one
1-[4-(difluoromethoxy)-2-methylphenyl]-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
1-{4-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-tert-butyl-4-({[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl](methyl)amino}methyl)pyrrolidin-2-one
N-(2-methoxyethyl)-1-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
3-fluoro-N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide