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7-(2,3-dihydro-1-benzofuran-5-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3,4-dimethoxy-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)benzene-1-sulfonamide
(2R)-2-amino-3-phenyl-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}piperidine-3-carboxamide
1-benzyl-3-methyl-4-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperazin-2-one
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl})amine
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1'-[(3-chloro-5-fluorophenyl)methyl]-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(furan-2-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(methylamino)pyridine-3-carboxamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{5-[2-(methylsulfanyl)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-chloro-6-methoxy-4-{[(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}phenol
3-(2-chlorophenyl)-N-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carboxamide
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
N-[2-(1H-indol-3-yl)ethyl]-4-methyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
3-[(2R,3R,6R)-5-(4-chlorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]pent-4-enamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(pyrazin-2-yl)ethyl]piperidin-2-one
8-{3-[1-(dimethylamino)ethyl]phenyl}quinolin-4-amine
1-(3-methylbutyl)-8-[1-(methylsulfanyl)propan-2-yl]-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,9aR)-3-(4-aminobutyl)-8-(2-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-methyl-1H-1,2,4-triazole
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
2-(dimethylamino)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(4-methylphenyl)acetamide
5-[1-(5-phenoxyfuran-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-9-oxo-N-(pyrazin-2-ylmethyl)-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
(R)-[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl](phenyl)methanol
{[(1R,5S,6S)-3-{[3-(furan-2-yl)phenyl]methyl}-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
4-benzyl-3-{2-[4-(ethanesulfonyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(3,4,5-trimethoxyphenyl)acetamide
7-(3-methoxypropyl)-2-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(2S)-1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]pyrrolidine-2-carboxamide
6-[(3S)-3-hydroxypyrrolidin-1-yl]-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
3-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propanamide
3-{[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]methyl}-1,2,3-oxadiazol-3-ium-5-olate
4-(piperidine-1-carbonyl)-2-[4-(1H-pyrazol-5-yl)phenyl]pyridine
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]acetamide
4-{[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
2-(2-cyclopropylpyrimidin-5-yl)-4-(3,3-dimethylpyrrolidine-1-carbonyl)-6-methylquinoline
N-[3-(4-fluorophenyl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxamide
3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-3-(oxan-4-yl)-6-(pyridine-3-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2H-1,3-benzodioxol-5-yl)-1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]propan-1-one
N-[2-(pyrazin-2-yl)ethyl]-2-(pyrrolidine-1-carbonyl)cyclohexane-1-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole