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3-amino-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
2-[4-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)-6-methylpyrimidin-2-yl]phenol
4-[4-oxo-7-(5-oxohexanoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
(4S,6R)-6-methyl-N-(2-methylpropyl)-2-sulfanylidene-N-(thiophen-3-ylmethyl)-1,3-diazinane-4-carboxamide
4-{[2-(ethylsulfanyl)ethyl]sulfamoyl}-N-[(3S)-pyrrolidin-3-yl]benzamide
3-methyl-N-{[1-(quinolin-8-ylmethyl)piperidin-3-yl]methyl}but-2-enamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[2-(3-methoxyphenyl)-1-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
7-(2,2-dimethylpropyl)-2-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
N-[4-methoxy-3-({[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]carbamoyl}amino)phenyl]acetamide
N,1-dimethyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-propyl-1H-pyrazole-5-carboxamide
2-{3-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]phenyl}-6-(4-methylphenyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
3-(1-ethyl-1H-imidazol-2-yl)-1-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperidine
[(2R)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl]methanol
N-[3-(1H-imidazol-1-yl)butyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-(1H-imidazol-1-ylmethyl)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-ol
5-[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]-N-phenylpyrimidin-2-amine
1-({1-[2-(1H-imidazol-5-yl)ethyl]-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl}methyl)-4-phenylpyrrolidin-2-one
3-(furan-2-yl)-3-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]propanoic acid
N,3,5,7-tetramethyl-N-(1-methylpyrrolidin-3-yl)-1H-indole-2-carboxamide
(2E)-N-[1-(5-{[(4-methoxyphenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-3-(thiophen-2-yl)prop-2-enamide
N-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
2-{4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]piperidin-1-yl}ethan-1-ol
8-(3-methylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2,3-dihydro-1-benzothiophene-2-carboxamide
3-[(2R,3R,6R)-5-[(3-methylthiophen-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-3-(ethylsulfanyl)propan-1-one
N-[4-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
2-{4-[2-(2-acetyl-4,5-dimethoxyphenyl)acetyl]morpholin-3-yl}acetic acid
3-{1-[(6-ethoxyquinolin-2-yl)methyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[(4-cyanophenyl)methyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
2-(1-methylpiperidin-2-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}acetamide
1-{[(3R,4R)-1-(3,5-difluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
(2S)-2-amino-1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-(1H-imidazol-4-yl)propan-1-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(1H-1,3-benzodiazol-1-yl)propanamide
6-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carbonitrile
2-{3-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]phenoxy}acetamide
1-(4-chloro-2-methoxy-5-methylphenyl)-3-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]urea
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-N-(propan-2-yl)pyridine-4-carboxamide
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidine
(3S,4S)-4-(3-methoxyphenyl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidin-3-ol
5-[1-(methoxymethyl)cyclobutyl]-3-(oxan-4-yl)-1-phenyl-1H-1,2,4-triazole
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
5-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-2,1,3-benzothiadiazole
8-[(3-hydroxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-({2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}methyl)piperidin-4-yl]methanesulfonamide
1-[2-(diethylamino)acetyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
5-[2-(benzyloxy)ethyl]-2-fluorobenzamide
6-[2-(morpholin-4-ylmethyl)phenyl]-1H-1,3-benzodiazole