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2-(6-chloro-2-oxo-2H-chromene-3-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[2-(4-methoxyphenyl)ethyl]-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-4-[4-({[(2,4-difluorophenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
2-amino-4-(1,2-dimethyl-1H-imidazol-5-yl)-6-(4-fluorophenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-3,4-dihydroquinazolin-4-one
6-cyclopropyl-2-(3-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
5-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-methyl-1,3-thiazole
6-[5-(2-ethylpyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]-2-methylheptan-2-ol
1-(3-chloro-2-methylbenzenesulfonyl)-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
6-(3,5-dimethoxyphenyl)-N-ethylpyridazin-3-amine
N-tert-butyl-2-(5,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)benzene-1-sulfonamide
3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-N-(3-methyl-1,2-thiazol-5-yl)benzamide
(2S,4R)-4-amino-N-ethyl-1-[(2-methoxynaphthalen-1-yl)methyl]pyrrolidine-2-carboxamide
8-(8-chloroquinolin-2-yl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N,5-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-6-methylpyridine-3-carboxamide
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-benzothiazole-5-carboxamide
methyl({[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
N-(2-benzylbutyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
6-methoxy-N-{3-[methyl(phenyl)amino]propyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[(3R,4S)-1-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-(butan-2-yl)-2,6-dioxo-N-(3-phenylprop-2-yn-1-yl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
6-(methoxymethyl)-2-[4-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-[(5-methylthiophen-2-yl)methyl]-3-(1H-pyrazol-4-yl)-N-(pyridin-2-ylmethyl)benzamide
2-(4-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}phenoxy)acetamide
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-N-(2-hydroxyethyl)-N-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(2-{1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-2-yl}ethyl)phenol
5-(2,3-dihydro-1H-inden-2-ylmethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-(4-{[2-(3-chlorophenyl)-8-methylquinolin-3-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
3-{1-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1-[3-(2-methylpyrimidin-4-yl)phenyl]urea
1-[4-chloro-2-(trifluoromethyl)phenyl]-3-ethyl-3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]urea
(3S,4S)-1-(2,6-dimethylquinoline-4-carbonyl)piperidine-3,4-diol
4-{[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-benzyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-chlorophenyl)-4-[4-(thiophen-2-yl)butanoyl]piperazin-2-one
(1S,5R)-6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-(5-methylfuran-2-yl)-N-[2-(propylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
(1S,5R)-3-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}propanamide
2-amino-6-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
4-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
1-(2-methoxybenzoyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylic acid
3-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}azetidin-3-yl)pyridine
1-ethyl-2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
4-(4-chlorophenyl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]butan-1-one
1-(1,4-dithiepan-6-yl)-4-[(2-fluorophenyl)methyl]piperidine
3-{[(3-hydroxypropyl)(propan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide