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1-[2-(2-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-6-methoxyphenoxy)ethyl]-1H-imidazole
(4S)-3-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-4-phenyl-1,3-oxazolidin-2-one
3-propoxy-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-1-carboxamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-(2-methoxyphenyl)propanamide
N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]pyridazine-4-carboxamide
[(1,4-dimethyl-1H-pyrazol-5-yl)methyl](furan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-[3-(azocan-1-yl)propanoyl]imidazolidin-4-one
ethyl 1-(1H-indol-2-ylmethyl)-4-(2-methoxyethyl)piperidine-4-carboxylate
4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methylpiperazin-2-one
2-[ethyl(pyridin-4-ylmethyl)amino]-2-(4-fluoro-3-methylphenyl)acetic acid
7-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(4-ethylphenyl)methyl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
N-[(3S,4R)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(1S,5R)-3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)(pyridin-2-ylmethyl)amine
2-(dimethylamino)-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-2-(3-methylphenyl)acetamide
7-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyridine-4-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[5-(propan-2-yl)thiophene-3-carbonyl]piperidin-4-ol
(2S)-3-(4-hydroxyphenyl)-2-{[3-(pyridin-4-yl)-1H-pyrazol-5-yl]formamido}propanamide
7-[(6-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(1-{[4-(methylsulfamoyl)phenyl]methyl}pyrrolidin-3-yl)methyl]acetamide
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-hydroxyethan-1-one
2-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]furan-3-carboxamide
5-ethyl-N-[(1-methylpiperidin-3-yl)methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-(4-{[(1-methylpiperidin-2-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-methyl-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-1-benzofuran-5-carboxamide
[(6-ethoxyquinolin-2-yl)methyl](methyl)(1H-pyrazol-3-ylmethyl)amine
5-{2-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(6-methoxypyrimidin-4-yl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-methyl-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-(3-phenylpropyl)pyrrolidin-3-yl]methanol
N3-butyl-N5-[2-(3-fluorophenyl)ethyl]-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(1,4-dioxan-2-ylmethyl)-15-methyl-13-oxo-9-(pyridin-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(2-hydroxy-4-methylbenzoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-1-[1-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-4-yl]piperidine-4-carboxamide
2-(3-methoxypropyl)-8-[2-(pyridin-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
3-[(2R,3R,6R)-5-(2-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-6-fluoro-3,4-dihydro-2H-1,4-benzoxazin-3-one
(2R)-2-amino-4-methyl-N-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]pentanamide
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(trifluoromethyl)benzamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(2-methylphenoxymethyl)piperidin-1-yl]ethan-1-one
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(pyridine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
[(3R,5R)-1-{[5-(2-fluorophenyl)furan-2-yl]methyl}-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
2-amino-4-(1H-imidazol-4-yl)-6-[1-(2-methoxyethyl)-1H-indol-3-yl]pyridine-3-carbonitrile
methyl 1-[(3S,5S)-1-[(4-fluorophenyl)methyl]-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-[(4-methanesulfonylphenyl)methyl]-1-methylpiperazine-2-carboxylic acid