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methyl[(1-methyl-1H-pyrazol-4-yl)methyl][(4-{[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-{imidazo[1,2-a]pyridin-2-ylmethyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{1-[2-(diethylamino)ethyl]-1H-imidazol-2-yl}benzoic acid
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
5-benzoyl-N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-methyl-6-{5-[(2R)-pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridazine
3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
1-[(5-acetylthiophen-3-yl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-[7-(hydroxymethyl)-9-(3-methoxypropyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-ol
5-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-methyl-N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-6-propylpyrimidin-4-amine
2-[3-chloro-5-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-4-carbonitrile
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]-4,4-difluoropiperidine
2-(carbamoylamino)-N-[(3R,4S)-1-[(dimethyl-1,3-thiazol-4-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
7-(cyclobutylmethyl)-2-(3-methylfuran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2,3-dihydro-1H-inden-2-yl)-N-[(2-methoxyquinolin-3-yl)methyl]piperidin-3-amine
8-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-methyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]pyrrolidine-3-carboxylic acid
3-[ethyl(pyridin-4-ylmethyl)amino]-N-(2-phenylethyl)piperidine-1-carboxamide
4-(2,5-dichlorophenyl)-6-methylpyrimidin-2-amine
6-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]pyridine-2-carboxylic acid
2,8-dimethyl-4-[4-(thian-4-yl)piperazine-1-carbonyl]quinoline
3-{[4-(3-chloro-4-fluorophenyl)piperazin-1-yl]methyl}piperidin-3-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-7-methyl-N-(pentan-3-yl)imidazo[1,2-a]pyridine-2-carboxamide
1-(cyclohexylmethyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-{1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
(3aS,6aS)-2-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(3R,4R)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
6-(3,4,5-trimethoxyphenyl)-1,3-benzothiazol-2-amine
(2R,3R,6R)-3-phenyl-5-(4-propylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[(3R,5R)-1-(4,6-dimethylpyrimidin-2-yl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
6-methoxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
2-fluoro-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
9-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
7-fluoro-3-{[(2-methoxyethyl)(propyl)amino]methyl}-1,2-dihydroquinolin-2-one
4-fluoro-N-(2-{[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethyl)benzamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
6-{[(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)amino]methyl}-1,4-oxazepan-6-ol
(3R,4R)-4-cyclobutyl-3-methyl-1-(2-methylpyridin-4-yl)piperidin-4-ol
2-cyclohexyl-6-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,3-benzoxazole
N-(oxolan-2-ylmethyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-[4-chloro-3-(trifluoromethyl)phenyl]-5-(methanesulfonylmethyl)pyridine
N-(1,3-thiazol-2-yl)-2-({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amino)propanamide
2-{3-[2-(dimethylamino)ethyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}pyrrolidine-1-carboxamide
3-methyl-8-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-cyclopropyl-4-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}pyrrolidin-2-one
1-(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one