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3-(2-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)cyclobutanecarboxamide
N,1,3-trimethyl-N-[1-(pyridin-2-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-cyclopropylpyrimidin-4-amine
N-{[1-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
2-methyl-6-[4-(pyridin-4-yl)piperazin-1-yl]pyrimidin-4-amine
N-(furan-3-ylmethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)-3-phenylpropan-1-ol
4-ethyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1,2,3-thiadiazole-5-carboxamide
N-(2-{1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}ethyl)acetamide
N,3-dimethyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}but-2-enamide
[1-({[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl](methyl)amino}methyl)cyclopentyl]methanol
1-(2-carbamoylethyl)-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1H-1,2,4-triazole-5-carboxamide
(3S,9aR)-8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3R,4R)-4-ethyl-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]piperidine-3,4-diol
1-(2-amino-4-{[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)but-3-en-1-one
2-(2,5-dimethoxyphenyl)-5-methyl-4-({2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-1,3-oxazole
4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxamide
3-[2-(2,6-dimethoxyphenoxy)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-(propane-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[(1R,2S)-2-phenylcyclopropyl]-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(1R,9aR)-1-({[2-(4-phenylpyrimidin-2-yl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
ethyl 1-[1-(ethoxycarbonyl)piperidin-4-yl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(3S)-2-oxoazepan-3-yl]-1,2-oxazole-3-carboxamide
N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-3-(1,2-oxazinan-2-yl)propanamide
(3R,4S)-4-cyclopropyl-1-[2-methoxy-5-(1H-pyrazol-1-yl)benzenesulfonyl]pyrrolidin-3-amine
1-(3-{[(6-hydroxy-6-methylheptan-2-yl)amino]methyl}-2,4,6-trimethylphenyl)ethan-1-one
(2-{furo[3,2-c]pyridin-4-yl}phenyl)methanol
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-{3-oxo-3-[2-(pyridin-3-yl)piperidin-1-yl]propyl}pyrrolidin-2-one
2-[1-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]phenol
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](4-methoxy-4-methylpentan-2-yl)amine
2-(dimethyl-1,3-thiazol-4-yl)-N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]acetamide
ethyl 3-({1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazol-4-yl}formamido)propanoate
2-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]pyridine-3-carbonitrile
3-({[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
N'-[2-(cyclohex-1-en-1-yl)ethyl]-N-[2-(methylsulfanyl)phenyl]butanediamide
3-[(3R,4S)-1-(2-methyl-2-phenylpropanoyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-[1-(1H-pyrazol-1-yl)propan-2-yl]-3,4-dihydro-2H-1-benzopyran-6-carboxamide
{3-[(2,4-difluorophenyl)methyl]-1-(6-methoxypyrimidin-4-yl)piperidin-3-yl}methanol
N,N-dimethyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-3,5-difluoropyridine-2-carboxamide
N-(8-methylquinolin-5-yl)-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl](methyl)[(3-methyloxetan-3-yl)methyl]amine
1-[(2-fluorophenyl)methyl]-N-[3-(methylsulfanyl)propyl]-1H-1,2,3-triazole-4-carboxamide
methyl 5-{[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylate
3-(4-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}phenyl)pyridine