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5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-3-(2-methylpropyl)-1,2-oxazole
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
N-(oxolan-2-ylmethyl)-2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
ethyl 3-{[2-(3-methoxyphenyl)piperidine-1-carbonyl]amino}propanoate
(3S,4S)-4-(dimethylamino)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-3-ol
4-[3-(2,6-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]morpholine
2-methyl-9-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
1-[4-(1H-pyrazol-3-yl)benzoyl]-4-(pyrrolidine-1-carbonyl)piperidine
[1-(2-methyl-1,3-thiazol-4-yl)ethyl][(5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazol-3-yl}furan-2-yl)methyl]amine
2-[(2-{ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}phenyl)amino]acetic acid
2-{4-[methyl({[2-(1H-pyrazol-1-yl)phenyl]methyl})amino]pyrimidin-5-yl}acetic acid
N-[2-(4-methylphenyl)propan-2-yl]-2-(2-oxocyclopentyl)acetamide
N-(3-methoxypropyl)-1-methyl-5-(5-methyl-1H-indole-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-[4-(hydroxymethyl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[4-(trifluoromethyl)phenyl]urea
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[4-(methylsulfanyl)benzoyl]piperidine
3-(2,5-dioxoimidazolidin-4-yl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}propanamide
(2S,4R)-1-benzyl-4-{[(3,4-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-[3-fluoro-5-(trifluoromethyl)phenyl]urea
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
8-[(2-chlorophenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-2-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]aniline
4-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-methyl-7-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl 3-(2-methylbenzamido)-6-[(3-methylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]acetamide
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
2-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-4-yl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-ethyl-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methyl-1H-pyrazole-5-carboxamide
2-{4-[3-fluoro-5-(propan-2-yloxy)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
2-(3-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenoxymethyl)pyridine
7-chloro-1-(2-phenoxyethyl)-3-({[2-(1H-1,2,4-triazol-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-(2-methoxyethyl)-9-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
8-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(1H-imidazol-1-ylmethyl)piperidine
N-[(2-propyl-1,3-thiazol-4-yl)methyl]-2,3-dihydro-1H-inden-2-amine
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[4-(pyrimidin-2-yloxy)piperidin-1-yl]acetamide
2-(propan-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidine-5-carboxamide
N-[(3R,5S)-1-cyclohexyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
2-(4-methylpiperidin-1-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
N-[3-(3-chlorophenyl)phenyl]-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
5-(methoxymethyl)-N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
(3S,4S)-4-(pyridin-2-yl)-1-(quinoxaline-6-carbonyl)pyrrolidine-3-carboxylic acid
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
4-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-2-methyl-1,3-thiazole
4-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
(2S,6S)-6-butyl-1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine