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N-(furan-2-ylmethyl)-N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}cyclohexanecarboxamide
1-[3-(3-methoxypropyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
4-[4-({3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)phenyl]-2-methylbut-3-yn-2-ol
5-{1-[(2,1,3-benzoxadiazol-5-ylmethyl)amino]ethyl}-N-cyclohexyl-N,4-dimethylpyrimidin-2-amine
7-(5-methylthiophen-2-yl)-4-(piperidin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(4-chloro-2-{[3-(hydroxymethyl)-4-methylpiperazin-1-yl]methyl}phenoxy)acetic acid
1-cyclohexyl-N3,N5-dimethyl-4-oxo-N3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
(1S,5R)-3-(1H-imidazol-4-ylmethyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
N,N-diethyl-4-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]aniline
(2S,4S)-4-amino-N,N-diethyl-1-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)pyrrolidine-2-carboxamide
1-{3-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]phenyl}imidazolidin-2-one
(3R,4R)-1-{[3-(furan-2-yl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
1-[4-(3-methoxyphenyl)phenyl]-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-amine
(2R,3S,6R)-5-{imidazo[1,2-b]pyridazine-3-carbonyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2,5-dioxoimidazolidin-1-yl)-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
methyl (2S,4S,5R)-5-(3-chlorophenyl)-1-methyl-4-[(2-methylpropyl)carbamoyl]pyrrolidine-2-carboxylate
1-[3-(2-ethylphenoxy)azetidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-3-carboxamide
3-methoxy-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-3-(1-methylpiperidin-3-yl)propanamide
3-benzyl-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazin-2-one
ethyl 3-({3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}amino)propanoate
methyl 6-[(4-ethoxyphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-hexyl-8-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(pyridin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}benzamide
3-cyclopropyl-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-1H-pyrazole-4-carboxamide
N-methyl-4-{[(3-methylthiophen-2-yl)methyl]amino}-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
2-cyclopropyl-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethan-1-one
4-ethyl-3-{1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(pyridin-2-yl)ethyl]acetamide
1-benzyl-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
1-cyclopentyl-6-oxo-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidine-3-carboxamide
1-{[4-(2-methylphenyl)phenyl]methyl}-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
3-{[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})carbamoyl}pyridin-1-ium-1-olate
({5-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-[4-(dimethylamino)phenyl]-3-{[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}propanamide
2-methyl-5-[(3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,2-oxazol-5-yl)methoxy]-1,3-benzothiazole
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-3-(pyridin-4-yl)propan-1-one
3-(4-methoxy-2-methylbenzoyl)-1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine
(1R,3R)-N1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}cyclopentane-1,3-diamine
2-{1,4-bis[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-{1-[1-(but-2-yn-1-yl)-1,2,3,6-tetrahydropyridin-4-yl]propan-2-yl}propanamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}quinoxalin-2-amine
(3S,4R)-1-(2-fluoro-5-methylbenzenesulfonyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
4-{[2-(dimethylamino)ethyl]amino}-5-methyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-phenyl-5-[2-(pyrrolidin-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(1H-indazol-1-yl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide