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2-(1-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
9-[2-(morpholin-2-yl)acetyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-benzyl-4-(pyrazine-2-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
6-methyl-2-({[3-(methylsulfanyl)propyl]amino}methyl)quinolin-4-ol
4-ethyl-1-(3-phenylpropyl)-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridazine
1-methyl-3-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1-[3-(oxolan-2-yl)propyl]urea
3-chloro-N-(2-methoxyethyl)-4-{[1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]oxy}benzamide
4-[(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-phenylethan-1-one
2-methyl-9-[3-(methylsulfanyl)propanoyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-[2-(3,5-difluorophenyl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]acetamide
4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
(2S,4S)-4-benzamido-N,N-diethyl-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
methyl 2-[4-(2-methoxyquinoline-4-carbonyl)-2-oxopiperazin-1-yl]acetate
2-(6-chloro-1,3-benzothiazol-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)benzonitrile
1-[(2S)-2-hydroxy-2-phenylacetyl]-4-phenoxypiperidine-4-carboxylic acid
1-(2-methylphenyl)-4-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]piperazine
8-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[2-(1H-imidazol-1-yl)propanoyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
8-(6-aminopyrimidin-4-yl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(4-{[(1-benzothiophen-2-ylmethyl)amino]methyl}phenoxy)-3-[benzyl(methyl)amino]propan-2-ol
3-[5-(quinoline-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-butyl-7-[(oxolan-2-ylmethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-[5-(oxan-2-yl)furan-2-yl]-1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-imidazole
2-methyl-5-phenyl-N-[1-(pyridin-3-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
(2S,4R)-4-amino-1-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-N-methylpyrrolidine-2-carboxamide
8-methyl-2-propyl-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,8-diazaspiro[4.5]decane
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-acetyl-8-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(2,3-dihydro-1H-isoindole-2-carbonyl)-5,6-dimethyl-1,2-dihydropyridin-2-one
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[1-(2-methoxyphenyl)ethyl]methylamine
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-[(6-methylpyridin-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,4R)-4-(2-methylphenyl)-1-[2-(propylsulfanyl)acetyl]pyrrolidine-3-carboxylic acid
5,6,7-trimethoxy-3-[(2-methyl-3-oxopiperazin-1-yl)methyl]-1,2-dihydroquinolin-2-one
5-[2-(2-methoxyphenoxy)propan-2-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenylpiperidine
(3S,4R)-1-[(dimethylcarbamoyl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
N-[2-(2-fluorophenyl)ethyl]-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(2,2-dimethylpropyl)-4-{[(2-phenyl-1,3-oxazol-4-yl)methyl]amino}pyrrolidin-2-one
1-(3-methylpyridin-4-yl)-4-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1,4-diazepane
1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-[3-(4H-1,2,4-triazol-4-yl)propyl]piperidin-4-amine
1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine