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5-{[3-(2-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-N-propylpyrimidin-2-amine
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(piperidin-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(5-{[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
2-methyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-(furan-2-ylmethyl)-5-methyl-6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]thieno[2,3-d]pyrimidin-4-amine
(2S,4S)-1-[(2-aminopyridin-3-yl)methyl]-4-(2-cyclopentylacetamido)-N-ethylpyrrolidine-2-carboxamide
2-methyl-6-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
N-{2-[1-(1-carbamoylethyl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}-3-cyanobenzamide
1-[7-methyl-3-(thiomorpholin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]azepane
4-{2-azaspiro[4.4]nonane-2-carbonyl}-7,8-dimethyl-2-(pyrimidin-5-yl)quinoline
methyl(pyridin-3-ylmethyl)[2-(1,3-thiazol-2-yloxy)hex-5-en-1-yl]amine
[3-(3-methylbut-2-en-1-yl)-1-(thiophene-2-carbonyl)piperidin-3-yl]methanol
4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
(1S,6R)-9-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-3,9-diazabicyclo[4.2.1]nonane
4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-{2-[(4-methoxyphenyl)sulfanyl]ethyl}-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
N-[(3-fluorophenyl)methyl]-6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-{[1-(carbamoylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-3-methoxybenzamide
2-[4-(4-fluorophenyl)-2-{[3-(hydroxymethyl)morpholin-4-yl]methyl}phenoxy]acetic acid
4-[1-(3-hydroxyphenyl)-5-oxopyrrolidine-3-carbonyl]-1-phenylpiperazin-2-one
2-[(2-amino-6-methylpyrimidin-4-yl)amino]-1-[2-(trifluoromethyl)phenyl]ethan-1-ol
1-{3-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]benzenesulfonyl}-1,4-diazepane
1-[4-(2-amino-5-methylpyrimidin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
1-methyl-3-[4-(2-methylphenoxy)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
4-ethyl-3-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N,6-dimethyl-2-propyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
(1S,5R)-6-(3,5-difluoropyridine-2-carbonyl)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane
5-[1-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-hydroxy-2-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}quinoline-6-carboxamide
3-{5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-ylmethyl]thiophen-2-yl}prop-2-yn-1-ol
N-methyl-N-(2-phenoxyethyl)-4-(piperidin-3-ylmethyl)benzamide
4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-N-(4-methylpyridin-2-yl)-4-oxobutanamide
(2S,4R)-4-amino-N-ethyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]pyrrolidine-2-carboxamide
(2S,4R)-N,N-diethyl-4-{2-[4-(hydroxymethyl)phenyl]acetamido}-1-methylpyrrolidine-2-carboxamide
1-amino-N-[(1-methylpyrrolidin-3-yl)methyl]cyclobutane-1-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-2,3-dihydro-1H-indene-2-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[4-methyl-6-(methylsulfanyl)quinolin-2-yl]pyrrolidin-3-yl]methanol
2-[4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
2-methyl-6-{1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidin-3-yl}pyrimidin-4-ol
(2S,4S)-4-{[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]amino}-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-4-[4-(pyrrolidine-1-sulfonyl)-1,4-diazepane-1-carbonyl]-1,3-thiazol-2-amine
4,4,4-trifluoro-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]butan-1-one
6-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
(3E)-1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pent-3-en-1-one
N-(3,3-diphenylpropyl)-6-(pyrazine-2-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
[3-(cyclopropylmethyl)-1-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}piperidin-3-yl]methanol
1-cyclopentyl-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
1-(4-chloro-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)piperidine
4-(2-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-2-oxoethyl)-5-methyl-2,3-dihydro-1H-pyrazol-3-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide