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2-cyclohexyl-1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
1-(2-{4-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
5-(4-{[4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
7-(8-methoxy-2-methylquinolin-5-yl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yloxy)ethyl]acetamide
4-{[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]methyl}benzoic acid
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-3-(pyridin-4-yl)propanamide
1-{[2-(methylsulfanyl)phenyl]methyl}-4-(1H-pyrazol-3-yl)piperidine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(1H-1,2,4-triazol-3-yl)benzamide
2-{3-[4-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}-6-ethoxy-4-methylquinazoline
N-[1-(4-fluorophenyl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1'-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}spiro[indene-1,4'-piperidine]
4-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-2-amine
3-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-fluoroquinolin-4-ol
7-[5-(hydroxymethyl)furan-2-carbonyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(3-chlorophenyl)methyl]-3-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]propanamide
2-[3-(3-methylphenyl)piperidine-1-carbonyl]phenol
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-3-(1H-pyrazol-1-yl)benzamide
2-(3-{[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]methyl}piperidin-1-yl)ethan-1-ol
5-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-2-cyclohexylpyrimidine
3-fluoro-N-{[7-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
3-methyl-8-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-methyl-7-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-(6-hydroxy-6-methylheptan-2-yl)-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(4-acetylphenoxy)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
[(4aS,8aR)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(6-methylpyridazin-3-yl)-decahydro-1,6-naphthyridin-4a-yl]methanol
2-{2-[(3,4-dimethoxyphenyl)methyl]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-[1-(1-phenylcyclopentanecarbonyl)piperidin-4-yl]methanesulfonamide
(2S,4S)-1-benzyl-4-{[(2,4-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(4,6-dimethyl-2-oxo-2H-pyran-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
5-({[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl](propan-2-yl)amino}methyl)pyrrolidin-2-one
(3S,5R)-N3-(6-methylpyridin-3-yl)-N5-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-3,5-dicarboxamide
8-(2-hydroxypyridine-3-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 4-({4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}methyl)thiophene-2-carboxylate
2-methyl-4-[5-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)thiophen-2-yl]but-3-yn-2-ol
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)(2-methylpropyl)(pyridin-2-ylmethyl)amine
7-(cyclobutylmethyl)-2-(1,4-dithiepan-6-yl)-2,7-diazaspiro[4.5]decane
[(2S)-1-[8-chloro-2-(furan-2-yl)quinoline-4-carbonyl]pyrrolidin-2-yl]methanol
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(2-hydroxyethyl)piperidin-4-yl]methyl}acetamide
1-methyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}piperidine-2-carboxamide
(3S,4R)-1-[(1-methyl-1H-indol-3-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
2-(2-phenyl-1H-imidazol-1-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
{1-[1-(cyclohexylmethyl)piperidin-3-yl]piperidin-4-yl}methanol
4-[1-(7-fluoroquinazolin-4-yl)piperidin-4-yl]pyrimidin-2-amine
3-[(2-oxopiperidin-3-yl)sulfamoyl]-N-(pyridin-3-yl)benzamide
1-cyclohexyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-4-carboxamide
2-[(propan-2-yl)amino]-N-[(4-sulfamoylphenyl)methyl]pyrimidine-5-carboxamide
6-tert-butyl-N-[2-(dimethylamino)pentyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine