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N-ethyl-5-(2-methoxyphenoxymethyl)-N-(oxan-4-yl)-1H-pyrazole-3-carboxamide
4-{2-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
methyl 4-{[(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amino]methyl}benzoate
methyl N-{4-[3-(propanamidomethyl)phenyl]phenyl}carbamate
3-{[1-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)pyrrolidin-3-yl]methyl}benzamide
N-(1-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N-[2-(2-hydroxyethoxy)ethyl]-4-(4-methoxyphenoxy)benzamide
1-(2-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
(1R,5R)-6-[(2-chloro-4-fluorophenyl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-methyl-8-[4-(piperidin-1-ylmethyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-(1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
6-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N4-methyl-N4-(quinolin-5-ylmethyl)pyrimidine-4,6-diamine
3-methyl-N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-5,6-dihydro-1,4-dioxine-2-carboxamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-N'-(2-methylphenyl)propanediamide
3-({methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]amino}methyl)pyridin-2-amine
6-ethyl-1,5-dimethyl-3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
4-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}-2,6-dimethylphenol
ethyl 1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-(4-acetyl-1,4-diazepan-1-yl)-2-(2,4-dimethoxyphenyl)acetic acid
1-(carbamoylmethyl)-N-[3-(4-chlorophenyl)propyl]piperidine-3-carboxamide
1-(morpholine-4-carbonyl)-4-(9H-purin-6-yl)-1,4-diazepan-6-ol
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[5-(propan-2-ylsulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
3-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(quinoline-8-carbonyl)piperidin-3-yl]propan-1-ol
2-(dimethylamino)-2-(2-fluorophenyl)-1-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
N-cyclopropyl-5-[(2,6-difluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,5,6-trimethylpyrimidin-4-amine
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(3-fluorophenyl)ethan-1-one
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[1-(3,5-difluorophenyl)cyclopropyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
4-[(3-fluorophenyl)methyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)-3-oxopiperazine-1-carboxamide
3-[2-amino-4-({1-azabicyclo[2.2.2]octan-3-yl}amino)-6-methylpyrimidin-5-yl]propanoic acid
9-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-(4-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
5-(2-phenylpyrrolidine-1-carbonyl)-2-(pyrrolidin-1-yl)pyrimidine
3-methoxy-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-2,3-dihydro-1-benzofuran-2-carboxamide
8-[1-(methylsulfanyl)propan-2-yl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N3-[3-(4-fluorophenyl)propyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-4-(1H-1,2,4-triazol-1-yl)aniline
(3S,4R)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
[2-(2-ethoxyphenoxy)ethyl](1H-imidazol-4-ylmethyl)methylamine
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(2-phenylethyl)piperazin-2-yl]ethan-1-ol
1-(2,2-dimethylpropyl)-4-{[(2E)-2-methylbut-2-en-1-yl]amino}pyrrolidin-2-one
N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-1-phenylmethanesulfonamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-methoxyethoxy)acetamide
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-2-(1H-1,2,4-triazol-1-yl)acetamide